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2-(2-hydroxyethyl)-8-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
(4aR,7aS)-1-methyl-4-(2-phenylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
1-[3-(cyclohexyloxy)-2-hydroxypropyl]-3-[3-(4H-1,2,4-triazol-4-yl)phenyl]urea
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
5-methyl-3-[2-(morpholin-4-yl)ethyl]-5-{1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-4-yl}imidazolidine-2,4-dione
(3R,9aR)-8-[(2-chlorophenyl)methyl]-3-[(1S)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-5-propyl-N-(quinoxalin-6-ylmethyl)-1,2-oxazole-3-carboxamide
N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1H-1,2,3-triazole-5-carboxamide
3-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-N-ethylpropanamide
methyl 3-(2,3-dihydro-1-benzofuran-5-ylmethyl)-9-[2-(2-fluorophenyl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1R,2S)-N-tert-butyl-2-(4-methyl-1,4-diazepane-1-carbonyl)cyclohexane-1-carboxamide
3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-methyl-1-[(5-propyl-1H-pyrazol-3-yl)methyl]urea
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[1-(carbamoylmethyl)-1H-imidazol-2-yl]-N-(2-ethoxyphenyl)piperidine-1-carboxamide
N-{2-[7-(1-benzofuran-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-(4-fluorophenyl)acetamide
1-ethyl-4-{[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
3-({[4-(3-fluorophenyl)oxan-4-yl]methyl}amino)-N-(1,3-thiazol-2-yl)propanamide
N-(diphenylmethyl)-2-(1-methyl-3-oxopiperazin-2-yl)acetamide
N,N-diethyl-1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]pyrrolidin-3-amine
2-(2H-1,2,3-benzotriazol-2-yl)-1-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]ethan-1-one
1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-2-(3-methyl-1H-1,2,4-triazol-5-yl)ethan-1-one
4-[1-methyl-3-(pyridin-3-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-2,1,3-benzoxadiazole
N-[(2R,3R)-1'-{[4-(difluoromethoxy)phenyl]methyl}-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
1-{4-[({1-[(2-fluorophenyl)methyl]piperidin-3-yl}(methyl)amino)methyl]thiophen-2-yl}ethan-1-one
N'-(2-fluoro-5-methylphenyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]butanediamide
4-({3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-3-(2,5-dimethylphenyl)-1H-pyrazole
N-methyl-N-[2-(2-methylphenyl)-1-{1-[2-(morpholin-4-yl)propanoyl]piperidin-4-yl}ethyl]-2-(1H-pyrazol-1-yl)acetamide
N-({7-[2-(2-chlorophenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-fluorobenzamide
5-(5-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazol-3-yl)-1H-1,3-benzodiazole
4-[(2-methyl-1H-imidazol-1-yl)methyl]-1-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidine
4-{3-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]phenyl}phenol
N-[(7-{[5-(2-chlorophenyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-2-phenylacetamide
4-amino-N-butyl-N-cycloheptylpyridine-2-carboxamide
methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
4-(4-fluorophenyl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-oxobutanamide
N-(1-{7-[(4-ethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
propyl (4aR,7aS)-4-[(2-ethylphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
1-{4-[3-(4-phenylbenzoyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
2-(2-{5-[2-(5-methylfuran-2-yl)propyl]-4-phenyl-1H-imidazol-1-yl}ethyl)pyrazine
(2S)-2-hydroxy-4-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]butanoic acid
N-[2-(2-chlorophenyl)-1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
N-ethyl-4-hydroxy-N-(pyridin-4-ylmethyl)-2-(thiophen-2-yl)pyrimidine-5-carboxamide
N-(propan-2-yl)-3-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)propanamide
1-(difluoromethyl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-3-carboxamide
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-N-[4-(3-fluorophenyl)phenyl]piperidine-3-carboxamide
1-(2-aminoethyl)-N-[3-(azepan-1-yl)-2-hydroxypropyl]-1H-1,2,3-triazole-4-carboxamide
3-{[(5-methylthiophen-2-yl)methyl]({[4-(pyrimidin-5-yl)phenyl]methyl})amino}propan-1-ol
N-({8-[(2,3-dimethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)furan-2-carboxamide
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(2-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane