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N-(1-benzylpyrrolidin-3-yl)-3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]propanamide
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N,N-diethyl-1H-pyrazole-4-carboxamide
5-(methoxymethyl)-N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]furan-2-carboxamide
1-phenyl-4-[3-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]piperidine
N-(1-hydroxypropan-2-yl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
methyl 3-(2-methoxybenzamido)-5-(pent-4-enamidomethyl)benzoate
(1R,5R)-6-benzyl-3-(pyrrolidine-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{[(2R,5S)-5-[(1-methyl-1H-indol-5-yl)methyl]oxolan-2-yl]methyl}piperidine-4-carboxylic acid
ethyl 4-({[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}amino)piperidine-1-carboxylate
3-(1-phenylcyclopropyl)-5-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
1-{2-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}pyrrolidin-2-one
2-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-(2-phenylethyl)piperazin-2-yl)ethan-1-ol
N-benzyl-3-{[3-(dimethylamino)pyrrolidin-1-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
7-fluoro-4-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-1,2-dihydroquinolin-2-one
ethyl 4-{6-[2-(2-chlorophenoxy)acetyl]-6-azaspiro[2.5]octane-1-carbonyl}piperazine-1-carboxylate
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(piperidin-1-yl)acetamide
methyl 3-[(2,3-difluorophenyl)methyl]-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(diethylsulfamoyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
2-[4-(2-methoxypyridin-3-yl)-1H-pyrazol-1-yl]-N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)acetamide
8-[(3,4-difluorophenyl)methyl]-1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 2-[(3-methyl-5-propyl-1-benzofuran-2-yl)formamido]-4-(methylsulfanyl)butanoate
N-(2-methoxyethyl)-N-[(3-methoxyphenyl)methyl]-4,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(3S,5R)-5-[4-(2-hydroxyethyl)piperazine-1-carbonyl]-N-(4-methylphenyl)piperidine-3-carboxamide
3-(4-chlorophenyl)-N-[2-(morpholin-4-yl)ethyl]-3-phenylpropanamide
4-[4-benzyl-4-(hydroxymethyl)piperidine-1-carbonyl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
3-ethyl-5-[2-(methylsulfanyl)ethyl]-1-(2-phenylethyl)-1H-1,2,4-triazole
5,6-dimethyl-2-oxo-N-[2-(2-propoxyphenyl)ethyl]-1,2-dihydropyridine-3-carboxamide
4-(3-methyl-3-phenylpiperidine-1-carbonyl)morpholine
7-(5-methylthiophen-2-yl)-4-(piperidine-1-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[(4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)methyl]-2,1,3-benzoxadiazole
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
4-[1-(4-chlorobenzoyl)piperidin-3-yl]-2-methyl-5-(3-methylphenyl)pyrimidine
3-[(2-cyclopropyl-1,3-benzoxazol-5-yl)methyl]-1λ6-thiane-1,1-dione
1-[(4-fluorophenyl)methyl]-4-methanesulfonyl-2-(propan-2-yl)-1,4-diazepane
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-ethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
2-(2,4-dichlorophenoxy)-N-[2-(1H-pyrrol-1-yl)ethyl]acetamide
4-[1-(1-methoxypropan-2-yl)-1H-imidazol-2-yl]benzoic acid
6-[2-(2-chloro-4-fluorophenyl)acetyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-[1-(furan-3-ylmethyl)-4-hydroxypiperidin-4-yl]-1-benzofuran-2-carboxamide
1-(2-methyl-4-{[3-(4-methyl-1,3-thiazol-5-yl)propyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(methylamino)-1,3-thiazole-4-carboxamide
4-[5-(2-aminoethyl)-2-methoxyphenyl]-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N3-methyl-N5-(2-methylpropyl)-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
2,6,8-trimethyl-N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]quinoline-4-carboxamide
3-(2-methoxyethyl)-5-[1-(2-phenylethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazole
6-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-5-chloropyridine-3-carboxylic acid
2-(cyclopropylmethyl)-9-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(5-methylpyridin-2-yl)-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-4-ol
8-[2-(methylamino)acetyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one