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4-(4-{[5-(3-chlorophenyl)furan-2-yl]methyl}piperazin-1-yl)-2-(3-methoxypropyl)-2,3-dihydro-1H-isoindole-1,3-dione
{3-[(2,4-difluorophenyl)methyl]-1-(thian-4-yl)piperidin-3-yl}methanol
(4aS,8aR)-6-[4-(aminomethyl)benzoyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
ethyl 5-{2-amino-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-2,4-dimethyl-1H-pyrrole-3-carboxylate
1-({1-[1-(methoxymethyl)cyclobutanecarbonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
1-[4-(furan-2-yl)benzoyl]-4-(4-methoxyphenyl)-2-methylpiperazine
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-cycloheptyl-5-[(dimethylsulfamoyl)amino]-1-methyl-2-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
5-(3-phenoxypropyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
2-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]pyridine-4-carboxamide
2-oxo-N-(2-phenylphenyl)-1,3-dioxa-8-azaspiro[4.5]decane-8-carboxamide
methyl 2-(2-{[2-(dimethyl-1,2-oxazol-4-yl)acetamido]methyl}-5-methyl-2,3-dihydro-1-benzofuran-7-yl)benzoate
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-8-fluoro-N-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
6-[(diethylamino)methyl]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
5-(2-methylphenyl)-3-(3-phenylpiperidin-1-yl)-1,2,4-triazine
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-propylfuran-2-yl)methyl]piperidine
N-({7-[(2E)-3-(2,5-difluorophenyl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-benzothiazole-2-carboxamide
4-cyclopentyl-3-(furan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-({[(dimethyl-1,2-oxazol-4-yl)methyl]amino}methyl)-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
1-benzyl-N5-cyclopropyl-N3-methyl-4-oxo-N3-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-(4-chlorophenyl)-3-[1-(3-methoxypropanoyl)piperidin-3-yl]propanamide
N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-(1-methylcyclopropyl)propanamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-[(pyridin-2-ylmethyl)amino]pyrrolidine-2-carboxamide
1-butanoyl-N-[3-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
(2S,4S)-4-amino-1-[2-(4-ethoxyphenyl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(1S,5R)-6-benzyl-3-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,2R,4R)-N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
4-[(1-methyl-1H-imidazol-2-yl)methyl]-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-[(2-methylphenyl)sulfanyl]ethan-1-one
N-methyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
(2S,4R)-4-{[(2,6-difluorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
3-({1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
2-methoxy-5-({methyl[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]amino}methyl)phenol
7-methoxy-N,N-dimethyl-2-(1-propyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
(1R,5R)-6-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-(2-methylpropyl)-8-(5-oxo-2,5-dihydro-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl]piperidine-4-carboxamide
7-chloro-1-(2-phenoxyethyl)-3-({[1-(thiophen-2-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
3-butyl-1-methyl-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]piperazin-2-one
8-(1,3-benzothiazol-2-yl)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,8-diazaspiro[4.5]decane
ethyl 2-[1-({4-[4-(furan-2-carbonyl)piperazin-1-yl]quinazolin-2-yl}methyl)piperidin-2-yl]acetate
2-[methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]-N-[1-(4-methylphenyl)ethyl]acetamide
2-chloro-N-{2-[2-(thiophen-3-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}benzamide
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]({[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
5-(2,4-difluorophenoxymethyl)-N-[(6-hydroxypyrimidin-4-yl)methyl]-1H-pyrazole-3-carboxamide
8-(2-methoxyethyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-[(3-hydroxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one