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3-{[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}pyridin-2-amine
3-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
3-methoxy-N-methyl-4-[(1-methylpiperidin-4-yl)oxy]-N-(2,2,6,6-tetramethylpiperidin-4-yl)benzamide
8-{[5-(pyridin-2-yl)thiophen-2-yl]sulfonyl}-2,8-diazaspiro[4.5]decan-3-one
3-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}-6-(trifluoromethyl)pyridin-2-ol
1-(4-methylphenyl)-4-(1-propylpiperidin-4-yl)piperazine
N-(2-hydroxyethyl)-2-(2,5,7-trimethyl-1H-indol-3-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
ethyl 5-({8-methyl-2,8-diazaspiro[4.5]decan-2-yl}methyl)-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
2-cyclopropyl-9-(2-methoxyethyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-(aminomethyl)-N-[4-chloro-3-(propylcarbamoyl)phenyl]piperidine-1-carboxamide
4-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
1-[(3-chlorophenyl)methyl]-3-(2,5-difluorobenzoyl)piperidine
1-benzyl-8-[(2-chlorophenyl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-3-(furan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
4-{2,5-dimethyl-3-[1-(oxan-3-ylmethyl)-4-phenyl-1H-imidazol-5-yl]-1H-pyrrol-1-yl}-4H-1,2,4-triazole
methyl 3-acetamido-1-[2-(4-methoxyphenyl)ethyl]-5-[(4-methylpentan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-1,5-dimethyl-1H-pyrrole-2-carbonitrile
2-(4-methyl-1H-imidazol-5-yl)-1-(3-phenylpropyl)-1H-imidazole
4-[1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)piperidin-4-yl]pyridine
1-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propan-1-one
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]benzamide
5-{3-methyl-3,9-diazaspiro[5.6]dodecane-9-carbonyl}-2-(methylsulfanyl)-3,4-dihydropyrimidin-4-one
5-amino-4-chloro-N-({5,7-dimethylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-pyrazole-3-carboxamide
N-{1-[1-(3-cyclopentylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
3-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
N-(3-methyl-1-{7-[(2E)-2-methylbut-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)pyridine-3-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine-3-carboxylate
1-methyl-4-[(2S,4R)-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carbonyl]-1,4-diazepane
4-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]-1,2-dihydroisoquinolin-1-one
6-[(3-chloro-4-hydroxyphenyl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
6-oxo-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-ethyl-3-(2-methylpropyl)-N-[1-(6-methylpyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
N-({7-[3-(3-fluorophenyl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)oxane-4-carboxamide
N-(oxan-4-yl)-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-{[3-(2-ethylphenoxy)azetidin-1-yl]methyl}-2,6-dimethoxyphenol
1-(furan-2-ylmethyl)-4-(oxane-4-carbonyl)-1,4-diazepan-6-ol
2-methyl-5-({3-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)pyridine
6-(4-methoxynaphthalen-1-yl)pyridine-2-carboxamide
N-butyl-N-(furan-2-ylmethyl)-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
7-[(8-methoxy-2H-chromen-3-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-(3-methoxyphenyl)-6-methyl-4-[(4-oxo-4H-chromen-3-yl)methyl]piperazin-2-one
N-{[(2S,4S)-1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-4-fluoropyrrolidin-2-yl]methyl}pentanamide
N-(1-hydroxy-3-methylbutan-2-yl)-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
2-({[(3R,4R)-1-(3-chlorothiophene-2-carbonyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
(2S,4R)-4-amino-N,N-diethyl-1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidine-2-carboxamide
1-cyclohexyl-4-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-2-one
methyl[2-(4-methylphenoxy)ethyl]{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-(5-methylthiophen-2-yl)ethyl]acetamide
8-[2-(2,4-dichlorophenoxy)acetyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
6-(2,5-dimethylfuran-3-yl)-N-ethyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide