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1-(5-ethyl-2-methylpyrimidin-4-yl)-N-methyl-N-(quinolin-6-ylmethyl)piperidin-4-amine
3-[2-(2-fluorophenyl)ethyl]-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine
N,3,5,7-tetramethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-indole-2-carboxamide
N-({7-[3-(2-chlorophenyl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-2-yl)acetamide
1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
4-(benzyloxy)-1-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperidine
N-[2-(2-fluorophenyl)-1-[1-(2-phenoxyacetyl)piperidin-4-yl]ethyl]-N-methyl-3-(methylsulfanyl)propanamide
3-(2-methoxyethyl)-1-[(3-methylphenyl)methyl]-5-(1H-1,2,3-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(ethyl)methylamine
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
[5-({methyl[(1-phenylpyrrolidin-3-yl)methyl]amino}methyl)furan-2-yl]methanol
N-[2-(morpholin-4-ylmethyl)phenyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
7-(2-methoxyethyl)-2-{[3-(trifluoromethyl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-[4-(4-fluorophenoxy)piperidin-1-yl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
N-{1-[7-(3-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-phenylpropanamide
3-{[4-(2-oxopyrrolidin-1-yl)piperidin-1-yl]methyl}benzonitrile
1-[(cyclohexylmethyl)carbamoyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-4-fluorobenzamide
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)acetamide
2-{4-[(2-methylphenyl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
N-[1-(dimethylamino)propan-2-yl]-6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)piperidine-1-carboxamide
3-[(3-hydroxy-2,2-dimethylpropyl)amino]-1-(3-methylpiperidin-1-yl)propan-1-one
N-benzyl-2-[1-cyclopentyl-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(2-hydroxyethyl)acetamide
N-(3-fluoropyridin-2-yl)-2-phenyl-5,6,7,8-tetrahydroquinazolin-5-amine
2-(methylsulfanyl)-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
1-ethyl-N-(2-hydroxy-2-phenylethyl)-5-methyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-4-carboxamide
2-{4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(2-{4-[(3-chloropyridin-4-yl)methyl]piperazin-1-yl}quinolin-3-yl)methanol
3-(3-hydroxy-3-methylbutyl)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]benzamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-(2-fluorophenyl)pyrrolidine
N-[(3S,4R)-4-(propan-2-yl)-1-(3-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-3-yl]acetamide
1-methyl-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
3-chloro-N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-N-(pyridin-3-ylmethyl)benzamide
N-cyclopentyl-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-{5-[(3,4-dimethylpiperazin-1-yl)methyl]pyrimidin-2-yl}benzenesulfonamide
N-({1-[(3-acetylphenyl)methyl]piperidin-3-yl}methyl)-2-(2-methoxyphenoxy)acetamide
5-chloro-2-hydroxy-N-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}benzamide
3-(3,4-difluorophenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
dimethyl(2-{[(5-methylthiophen-2-yl)methyl]({[5-(oxan-2-yl)furan-2-yl]methyl})amino}ethyl)amine
4-{4-ethyl-6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidin-2-yl}morpholine
6-[2-(cyclohex-1-en-1-yl)acetyl]-N-[3-(pyridin-4-yl)propyl]-6-azaspiro[2.5]octane-1-carboxamide
6-methoxy-N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}pyrimidin-4-amine
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-(pyrazin-2-yl)propan-1-one
2-methyl-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
methyl (2S,4R)-1-[(3,4-difluorophenyl)methyl]-4-[2-(4-fluorophenyl)acetamido]pyrrolidine-2-carboxylate