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N-(3-hydroxy-2,2-dimethylpropyl)-3-(3-hydroxy-3-methylbutyl)benzamide
[5-(1-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-imidazol-2-yl)furan-2-yl]methanol
1-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-3-(piperidin-3-yl)benzamide
3-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[1-(4-methoxyphenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
2-(dimethylamino)-2-(3-fluorophenyl)-N-[(4-fluorophenyl)methyl]-N-(2-hydroxyethyl)acetamide
N-(4-methoxyphenyl)-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]propanamide
3-fluoro-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)benzamide
N,N-diethyl-1-[(1s,4s)-4-(2,3-dimethoxybenzamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-N-methylpyridin-2-amine
3-[4-({4-[3-(dimethylamino)-2-hydroxypropoxy]phenyl}methyl)piperazin-1-yl]-1,2-dihydropyrazin-2-one
4-ethoxy-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]pyrimidin-2-amine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-{[1-(2-hydroxyethyl)piperidin-4-yl]methyl}benzamide
N-[1-(7-{[5-(methoxymethyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-methylpropanamide
N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
5-[1-(2-ethylbutyl)piperidin-4-yl]-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
7-[(3,4-difluorophenyl)methyl]-2-[3-(methylsulfanyl)propyl]-2,7-diazaspiro[4.5]decan-6-one
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methylpropanamide
1-{1'-[2-(methylamino)pyridine-4-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
6-fluoro-2-(1-propyl-1H-pyrazol-4-yl)-4-(pyrrolidine-1-carbonyl)quinoline
1-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
dimethyl[1-(pyridin-2-yl)-2-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-1H-imidazol-1-yl]ethyl]amine
5-(methanesulfonylmethyl)-3-phenyl-1-[4-(propan-2-yl)phenyl]-1H-1,2,4-triazole
3-chloro-N-{[7-fluoro-5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-2-carboxamide
methyl (1R,3S,3aR,6aS)-1,5-diethyl-3-(5-fluoro-2-methoxyphenyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-{2-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-methyl-1'-[3-(methylsulfanyl)butyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
{[4-(butan-2-yloxy)-3-chloro-5-methoxyphenyl]methyl}(ethyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(2-oxo-2-phenylacetyl)pyrrolidin-3-yl]acetamide
2-(ethylamino)-N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methylpyrimidine-5-carboxamide
N-[2-(2-fluorophenyl)-1-[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-yl]ethyl]-N,2-dimethylfuran-3-carboxamide
1-benzyl-5-cyclopentyl-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{2-[(2-butyl-1H-imidazol-4-yl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}-2,2-dimethylpropan-1-one
8-[(2-methyl-1,3-oxazol-4-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
(2S)-2-({5-[(4-benzylpiperidin-1-yl)methyl]-1,2-oxazol-3-yl}formamido)propanamide
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl)[(3-fluoro-4-methoxyphenyl)methyl]amine
methyl 4-[({1-[2-(dimethylamino)ethyl]-6-oxopiperidin-3-yl}formamido)methyl]benzoate
7-methyl-3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-cyclobutyl-N-[1-(1H-indol-1-yl)propan-2-yl]-5-(2-methoxyacetamido)-1-methyl-1H-1,3-benzodiazole-7-carboxamide
1-ethyl-8-(1H-indol-2-ylmethyl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
4-cyclopentanecarbonyl-2-[(3-fluorophenyl)methyl]morpholine
N-benzyl-N-methyl-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
N-(adamantan-1-yl)-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,1,5-trimethyl-1H-pyrazole-3-carboxamide
5-[(4-chlorophenyl)methyl]-5-(3-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-3-oxopropyl)pyrrolidin-2-one
3-(5-methylfuran-2-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(pyrimidin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[(3R,4S)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid