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1-(2-methoxyethyl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]pyrrolidine-3-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-N-{1-[(3-methylphenyl)methyl]cyclopropyl}propanamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-(2,5-dioxoimidazolidin-4-yl)acetamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
1-{4-[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]piperidin-1-yl}ethan-1-one
N-methyl-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(quinolin-5-ylmethyl)propanamide
N-(1-{1-[2-(pyridin-2-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
4-({3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
(2S,4R)-4-amino-N-ethyl-1-[2-hydroxy-5-(1H-pyrrol-1-yl)benzoyl]pyrrolidine-2-carboxamide
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)[(6-methylpyridin-3-yl)methyl]amine
1-(2-methyl-1-benzofuran-5-carbonyl)-3-(2-methylphenyl)pyrrolidin-3-ol
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
6-({3-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)quinoline
2-{2-[1-(2-ethoxyethyl)-4-phenyl-1H-imidazol-5-yl]phenoxy}acetamide
2-{5-[2-(morpholin-4-ylmethyl)-1,4-oxazepane-4-carbonyl]-1H-pyrazol-3-yl}phenol
1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
2-methyl-5-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1H-1,3-benzodiazole
1-{4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]piperidin-1-yl}-2-methoxyethan-1-one
5-(2-chlorophenyl)-N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]furan-2-carboxamide
2-[({1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
2-chloro-6-fluoro-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
5-{2-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-1H-imidazol-1-yl}-2-methylpyridine
3-(5-methylpyridine-3-carbonyl)-3,9-diazaspiro[5.6]dodecan-10-one
1-(2,3-dimethylquinoxalin-6-yl)-3-methyl-3-[(5-propyl-1H-pyrazol-3-yl)methyl]urea
1-[(3-chlorophenyl)methyl]-1-methyl-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
4-(4-ethoxy-3-methylphenyl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}butanamide
N-cyclopropyl-N'-(2-fluoro-5-methylphenyl)-N-[(3-methylthiophen-2-yl)methyl]butanediamide
4-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}-N-(1,3-thiazol-2-yl)benzamide
N-[2-(propan-2-yl)-2H-1,2,3-triazol-4-yl]-2-{3-[2-(trifluoromethyl)phenyl]-1H-pyrazol-1-yl}acetamide
(1S,5R)-3-(2-aminopyridine-4-carbonyl)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(1H-imidazol-1-yl)-1-[(2-phenylethyl)carbamoyl]piperidine-4-carboxylic acid
5-methyl-N-[2-(4-methylmorpholin-2-yl)ethyl]-1-(pyridin-2-yl)-1H-pyrazole-4-carboxamide
(1S,4S)-5-(3,5-dimethylbenzoyl)-2-(2-methoxy-5-methylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
6-[(2,5-dimethoxyphenyl)methyl]-N-methyl-N-[2-(4-methylphenoxy)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
N-cyclopropyl-2-{[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]amino}acetamide
9-{9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(2,4-dimethoxyphenyl)methyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
1-[2-(1H-imidazol-2-yl)benzoyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
3-[4-(5-acetyl-4-methylpyrimidin-2-yl)piperazin-1-yl]-1λ6-thiolane-1,1-dione
(3R,4R)-3-cyclopropyl-1-(5-methoxyfuran-2-carbonyl)-4-methylpyrrolidin-3-ol
4-(azocan-1-yl)-N,N-bis(2-hydroxyethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
4-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]morpholine-2-carboxylic acid
5-methoxy-3-[(2-methyl-1H-indol-5-yl)methyl]-3,4-dihydroquinazolin-4-one
3-(2-methoxyethyl)-1-[2-(methylamino)pyridine-4-carbonyl]piperidine-3-carboxylic acid
N-(3-{2-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-2-oxoethoxy}phenyl)propanamide
benzyl({[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-cyclopentyl-2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-[4-({3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}methoxy)phenyl]ethan-1-one
2-(1-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane-6-carbonyl)-N,N-dimethylaniline
3,5,7-trimethyl-2-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidine-1-carbonyl}-1H-indole