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N-cyclopentyl-5-methoxy-N-[(2-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-2-carboxamide
N-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-N-methyloxolan-3-amine
2-(5-{2-[cyclohexyl(methyl)amino]pyridin-3-yl}-3-methyl-1H-1,2,4-triazol-1-yl)acetic acid
5-[1-(2,2-dimethylpropanoyl)piperidin-4-yl]-3-[(4-fluorophenyl)methyl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
3-{1-methyl-5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}-N-(4-methylphenyl)-3-oxopropanamide
5-[1-(cyclopropylmethyl)-1H-pyrazol-3-yl]-4-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3-thiazol-2-amine
2-cyclopropyl-4-methyl-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
N-(1-benzothiophen-5-ylmethyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
N-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-N-methyl-1-(2-phenylethyl)piperidin-3-amine
4-(2-{3-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxoethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
1-(benzyloxy)-8-[2-(2,6-difluorophenyl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
8-methoxy-2-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}quinoline
3-(3-methoxyphenyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[2-(2-chlorophenyl)ethyl]-5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)pyrrolidin-2-one
methyl 5-{[(4-fluorophenyl)methyl]amino}-3-(2-methoxyacetamido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-benzyl-N-butyl-1-[1,3-dioxo-2-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[1-(1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3,4,5-trimethoxybenzamide
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-N-(3,4-dimethylphenyl)piperidine-1-carboxamide
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2,3-difluorobenzamide
N-[(3R,4R)-1-[2-(3-fluorophenoxy)acetyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
N-[2-(1-ethylpiperidin-3-yl)ethyl]-5-(propan-2-yl)-1,3-oxazole-4-carboxamide
2-amino-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N,6-dimethylpyrimidine-4-carboxamide
2-[3-(3-acetylphenyl)phenoxy]acetamide
2-propyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1,3-thiazole-4-carboxamide
(2S,4S)-4-amino-1-[2-(4-chloro-3-methyl-1H-pyrazol-1-yl)acetyl]-N-ethylpyrrolidine-2-carboxamide
5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-N-[2-(thiophen-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-[1-(pyrazin-2-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
2-{2-[1-(3-fluoro-4-methoxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
1-[3-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]pyrrolidin-2-one
N-(4-methylpentan-2-yl)-1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
3-{[ethyl(methyl)amino]methyl}-3-hydroxy-1-[(3-methoxyphenyl)methyl]piperidin-2-one
5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]-N-[2-(pyrrolidin-1-yl)ethyl]pyridin-2-amine
[(4-chloro-2-fluorophenyl)methyl](methyl)[(3-methylpyridin-2-yl)methyl]amine
2-(2-{6-[(3-methoxyphenyl)methoxy]-3-oxo-4-(2-phenylethyl)-1,4-diazepan-1-yl}-2-oxoethyl)-4-methyl-1,2-dihydrophthalazin-1-one
(3R,4R)-3-methyl-1-(5-methylthiophene-3-carbonyl)-4-(oxan-4-yl)piperidin-4-ol
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(pyridin-2-ylsulfanyl)acetamide
5-{3-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]propanoyl}-N-cyclopropyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N'-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-N-propylethanediamide
3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridin-2-ylmethyl)piperidin-3-yl]-N-(3-methylphenyl)propanamide
2-{[benzyl(1,3-thiazol-2-ylmethyl)amino]methyl}-6-methylphenol
3-{[(butan-2-yl)(pyridin-3-ylmethyl)amino]methyl}-2-chloro-6-methoxyphenol
1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
6-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-1-methyl-3-phenyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-{1-[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-3-yl}propanamide
6-ethyl-2-oxo-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,2-dihydropyridine-4-carboxamide
2-[(2R,3R)-2-hydroxy-3-(pyrrolidin-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]pyridine-4-carbonitrile
1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(2-propoxyethyl)piperazine
7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-4-(oxolane-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-ethyl-3-methyl-N-[2-(1H-pyrrol-1-yl)ethyl]piperidine-3-carboxamide