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N-[2-(2,4-difluorophenyl)-1-{1-[(4-methylphenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
5-[1-(carbamoylmethyl)piperidine-3-carbonyl]-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
N-({7-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-fluorobenzamide
4-{2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-1-(4-methoxyphenyl)piperazin-2-one
3-(diphenylmethyl)-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-sulfonamide
[(4aS,8aR)-6-cyclopropanecarbonyl-1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-N'-(4-methylphenyl)propanediamide
[3-(2-phenylethyl)-1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-3-yl]methanol
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-(pyrazin-2-yl)ethan-1-one
[5-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-2-(propan-2-yloxy)phenyl]methanol
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]benzamide
{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}bis(prop-2-en-1-yl)amine
N-(4-methoxy-2-methylphenyl)-3-(4-phenylbenzoyl)piperidine-1-carboxamide
N-(2,2-dimethyloxan-4-yl)-1-(3-phenylphenyl)piperidin-4-amine
3-[2-(3,4-dimethylphenoxy)ethyl]-1-[4-(morpholin-4-ylmethyl)phenyl]urea
1-(4-fluorophenyl)-2,2-dimethyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]cyclopropane-1-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-5-ethyl-1,3-oxazole-4-carboxamide
2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]acetamide
methyl 5-(5-hydroxy-1,2-dimethyl-1H-indole-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
(3S,4S)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
4,6-dimethyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(5-ethyl-1,2-oxazole-3-carbonyl)-4-(furan-3-carbonyl)-1,4-diazepane
(2S,4R)-4-amino-1-(4-ethyl-5-methylthiophene-3-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-{benzyl[(4-methoxy-3,5-dimethylphenyl)carbamoyl]amino}propanamide
1-[(4-methoxyphenyl)methyl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N,N,7,8-tetramethyl-2-[2-(pyridin-3-yl)pyrimidin-5-yl]quinoline-4-carboxamide
1-{3-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}ethan-1-one
N-(2-hydroxybutyl)-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
(3S,4R)-1-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
methyl 4-[({1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazol-4-yl}formamido)methyl]benzoate
1-(2-methoxyphenyl)-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-1H-pyrazole-4-carboxamide
3-{2-[2-(cyclohexylmethyl)morpholin-4-yl]-2-oxoethyl}-1,2,3-oxadiazol-3-ium-5-olate
3-(3-chlorophenyl)-N-[2-(1H-imidazol-4-yl)ethyl]-3-phenylpropanamide
N-[(5-methylfuran-2-yl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(benzylcarbamoyl)-4-phenoxypiperidine-4-carboxylic acid
ethyl 2-[1-(1-cyclopropyl-6-oxopiperidine-3-amido)cyclohexyl]acetate
[(2,3-difluoro-6-methoxyphenyl)methyl](2-methoxyethyl)(oxolan-2-ylmethyl)amine
N-[(3S)-2-oxoazepan-3-yl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
(3aR,6aR)-2-[(2-fluoro-4-methoxyphenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[4-(1,4-diazepan-1-ylmethyl)phenyl]-6-(methoxymethyl)-3,4-dihydropyrimidin-4-one
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(2-methoxyethyl)methylamine
2-(dimethylamino)-2-(3-fluorophenyl)-N-[3-(pyridin-3-yloxy)propyl]acetamide
(3R,5S)-N-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-5-(piperidine-1-carbonyl)piperidine-3-carboxamide
1-[1-(3,4-difluorobenzoyl)piperidin-4-yl]-3-phenylpropan-1-ol
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]piperidine
2-(5-{[(cyclopropylmethyl)sulfanyl]methyl}-1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-3-yl)acetamide
3-({1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
2-(2H-1,3-benzodioxol-5-yl)-N-cyclopentyl-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)acetamide
4-[4-(2-ethoxyacetyl)-2-oxopiperazin-1-yl]benzonitrile
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methylpyrrolidine-3-carboxamide