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N-[3-(morpholin-4-yl)propyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-3-phenyl-N-[2-(1,3-thiazol-4-yl)ethyl]propanamide
6-[(3-methoxyphenyl)methoxy]-4-(4-methyl-1,3-oxazole-5-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
2-(methylsulfanyl)-3-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)pyridine
1-{2-[2-(2-methoxyphenyl)acetamido]ethyl}-N-phenyl-1H-1,2,3-triazole-4-carboxamide
methyl 6-(4-fluorobenzoyl)-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[4-(4-cyclopentylpiperazine-1-carbonyl)-5-methyl-1H-pyrazol-1-yl]-4-(2,5-dimethoxyphenyl)pyrimidine
4-{2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-oxoethyl}-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
2-(3-{[3-(hydroxymethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
N-cyclopropyl-3-[1-(1-phenylcyclohexanecarbonyl)piperidin-4-yl]propanamide
4-{5-methyl-4-[2-(2-methylphenoxy)acetyl]-2-oxopiperazin-1-yl}benzonitrile
N-(furan-2-ylmethyl)-3-({[(1R,2R)-2-hydroxycyclohexyl]methyl}amino)propanamide
methyl 3-(3-{[(2-chlorophenyl)formamido]methyl}piperidine-1-carbonyl)benzoate
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-5-methoxyfuran-2-carboxamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-methylbenzamide
4-[1-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)ethyl]morpholine
N-(butan-2-yl)-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-(pyridin-3-ylmethyl)benzamide
1-(2-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-2-oxoethyl)piperidin-2-one
(2S,4S,5R)-4-{[2-(1H-imidazol-1-yl)ethyl]carbamoyl}-1,2-dimethyl-5-phenylpyrrolidine-2-carboxylic acid
4-(5-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-[2-(4-methoxyphenyl)ethyl]acetamide
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-1-(4-hydroxy-4-phenylpiperidin-1-yl)ethan-1-one
2-methyl-6-({4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
(1r,4r)-4-{[2-(2,4,7-trimethyl-1H-indol-3-yl)acetamido]methyl}cyclohexane-1-carboxylic acid
4-[(2,3-dimethoxyphenyl)methyl]-5-methyl-1-(2-methylphenyl)piperazin-2-one
(3aS,6aR)-3-[3-(4-methoxyphenyl)propyl]-5-(oxan-4-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(2R,4R,6S)-2-tert-butyl-6-(1,4-dimethylpiperidin-4-yl)oxan-4-yl]acetamide
1-{1-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]piperidin-4-yl}piperidin-3-ol
2-(dimethylamino)-4-methyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]pyrimidine-5-carboxamide
5-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
N-{[4-hydroxy-1-(1-methyl-1H-pyrazole-4-carbonyl)azepan-4-yl]methyl}-2-(thiophen-2-yl)acetamide
N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
4-chloro-1-ethyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1H-pyrazole-3-carboxamide
1-[3-(phenylamino)piperidin-1-yl]-2-(1-propylpiperidin-4-yl)ethan-1-one
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
2-(3-chloro-4-hydroxyphenyl)-1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
1-{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-2-yl)piperazine
methyl (1R,3S,3aR,6aS)-3-(4-hydroxy-2-methoxyphenyl)-5-methyl-1-(2-methylpropyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-N-(1,3-thiazol-2-yl)propanamide
(1S,9S)-11-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
4-({4-[3-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]furan-2-yl}methyl)morpholine
1-[benzyl(methyl)amino]-3-(4-{[methyl(pyridin-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
N-methyl-2-(methylsulfanyl)-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
N-ethyl-N-(pyridin-4-ylmethyl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
2-({[2-(methylamino)pyridin-3-yl]methyl}({[4-(methylsulfanyl)phenyl]methyl})amino)ethan-1-ol
4-(2,6-dimethylpyrimidine-4-carbonyl)-2-(2-methoxyethyl)morpholine
4-hydroxy-N-methyl-2-(4-methylphenyl)-N-(2-phenoxyethyl)pyrimidine-5-carboxamide
1-[cyclohexyl(methyl)amino]-3-[2-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-5-methyl-1,2-oxazole-3-carboxamide
methyl 2-{[5-(4-fluorophenyl)-4-[1-(furan-2-carbonyl)piperidin-3-yl]pyrimidin-2-yl]sulfanyl}acetate