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N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
3-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridine
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
3-(4-methoxyphenyl)-N-methyl-3-phenyl-N-[2-(1H-pyrazol-1-yl)ethyl]propanamide
3-[(3-fluorophenyl)methyl]-N-{[3-(trifluoromethoxy)phenyl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
3-[(3-ethoxyphenyl)methyl]-9-methoxy-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3R,9aR)-3-[(1S)-1-hydroxyethyl]-8-(quinolin-8-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[(2R,3R)-2-hydroxy-1'-(1-methyl-1H-pyrrole-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]piperazin-2-one
methyl 4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-4-oxobutanoate
5-fluoro-2-[1-(pyrrolidine-1-carbonyl)piperidin-2-yl]-1H-1,3-benzodiazole
N-{[7-(3-phenylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine-4-carboxamide
1-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-6-azaspiro[2.5]octane
1-(5-{[ethyl(2-methylprop-2-en-1-yl)amino]methyl}-2-methoxyphenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
1-[3-(azepan-1-ylmethyl)phenoxy]-3-(4-ethylpiperazin-1-yl)propan-2-ol
N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-2-(oxan-2-ylmethoxy)acetamide
2-{3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-1-methylpiperidine
1-(cyclopropylmethyl)-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-2-(propan-2-yl)-1,4-diazepane
1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
4-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]-1-(propan-2-yl)pyrrolidin-2-one
4-(4-chlorophenyl)-N-[2-(1H-imidazol-1-yl)propyl]butanamide
1-(piperidin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
methyl 5-{2-[4-(propan-2-yl)morpholin-2-yl]acetyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-(2-{7-[(2-chloro-6-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
2-methyl-1-[2-(2,3,6-trimethylphenoxy)acetyl]-1,4-diazepan-5-one
1-[4-({4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
N4-[cyclopropyl(6-methylpyridin-2-yl)methyl]-N2,N2-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
7-(cyclobutylmethyl)-2-[(4-fluoro-3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
3-[2-(3,3-diethylpyrrolidin-1-yl)-2-oxoethyl]-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-2-(furan-2-yl)-2-oxo-N-(oxolan-2-ylmethyl)acetamide
1-methyl-4-{[1-(2-phenylethyl)-5-(2H-1,2,3-triazol-2-ylmethyl)-1H-1,2,4-triazol-3-yl]methyl}piperidine
2-(piperidine-1-carbonyl)-3-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrazine
(3S,4S)-4-(pyrrolidin-1-yl)-1-(quinolin-4-ylmethyl)pyrrolidin-3-ol
N-[3-(1H-indol-2-yl)phenyl]-1-{spiro[2.3]hexane-1-carbonyl}piperidine-4-carboxamide
1-benzyl-N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
(1H-imidazol-2-ylmethyl)(methyl)[(2-phenylphenyl)methyl]amine
4-[5-({3-[benzyl(methyl)amino]piperidin-1-yl}methyl)thiophen-2-yl]-2-methylbut-3-yn-2-ol
4-(3-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}propyl)piperazin-2-one
5-(1H-indol-1-ylmethyl)-N-methyl-N-[(5-methylthiophen-2-yl)methyl]-1H-pyrazole-3-carboxamide
methyl (2S,4R)-1-methyl-4-(1-methyl-1H-imidazole-4-sulfonamido)pyrrolidine-2-carboxylate
1-[2-(4-chlorophenyl)ethyl]-N-methyl-6-oxo-N-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
methyl 1-{[4-(furan-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-4-carboxylate
N-(1-{4-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]phenyl}ethyl)acetamide
1-[(4-methoxypiperidin-1-yl)sulfonyl]-3-methyl-3-phenylpiperidine
4-{1-[4-(1H-1,2,3,4-tetrazol-5-yloxy)phenyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
N-cyclopentyl-1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]pyrrolidin-3-yl]methanol
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
2-[1-(3-methylbutyl)-4-[(4-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
4-chloro-1,5-dimethyl-N-{1-[2-(trifluoromethyl)phenyl]ethyl}-1H-pyrazole-3-carboxamide
N-[2-(3-methoxyphenyl)-1-{1-[(8-methoxyquinolin-2-yl)methyl]piperidin-4-yl}ethyl]-N-methylcyclopropanecarboxamide