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3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-8-(2-methylpyrimidin-4-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]acetamide
5-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-2-phenylfuran-3-carboxamide
(2S)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(6-methoxynaphthalen-2-yl)propanamide
1-(3-chlorophenyl)-2-(cyclopent-1-ene-1-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-(5-chloro-2-methylphenyl)-N'-[(5-methylpyrazin-2-yl)methyl]propanediamide
2-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)pyridine-3-carboxylic acid
(2E)-N-({8-cyclopropanecarbonyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-3-(3,5-difluorophenyl)prop-2-enamide
1,9-dimethyl-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[3-(1H-pyrazol-1-yl)propyl]amine
2-ethyl-1-{2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}-1H-imidazole
3-[(benzylamino)methyl]-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
2-(2-{[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-cyclohexyl-3-({[2-(trifluoromethoxy)phenyl]carbamoyl}amino)propanamide
6-methyl-5-[5-(4-methyl-1H-imidazol-2-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
3-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-1-(quinolin-7-yl)urea
2-[2-ethoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]quinoxaline
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methyl-1H-indole-2-carboxamide
6-cyano-N-[4-(2,2-dimethylpropanamido)-3-methylphenyl]pyridine-3-carboxamide
1-[5-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
N-cyclopentyl-N-({4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)cyclohexanecarboxamide
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-(naphthalene-2-carbonyl)piperidine
2-{1-[(4-fluorophenyl)methyl]-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-2-yl}ethan-1-ol
(2S,4R)-1-[(2-methoxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-fluoro-4-methoxy-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]benzamide
2-(cyclopent-2-en-1-yl)-1-[4-({4-[(methylamino)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidin-1-yl]ethan-1-one
7-(cyclopropylmethyl)-2-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
3-[5-(4-methyl-1H-imidazole-5-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-3-ol
6-(3-chlorophenyl)-7-(cyclopropylmethyl)-N-(2-methoxyethyl)-N-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-{1-propyl-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl}-1H-indole
2-(2-{3-cyclohexyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-oxoethyl)-4-methyl-1,2-dihydrophthalazin-1-one
N-(3-benzylphenyl)-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-3-(3-methylphenoxymethyl)piperidine
2-(4-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
3-{[1-(5-cyclopropyl-4-phenyl-1H-imidazol-1-yl)propan-2-yl]oxy}pyridine
N-(5-chloro-2-methoxyphenyl)-3-[1-(2-phenylethyl)piperidin-3-yl]propanamide
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(2-methylphenyl)propanamide
4-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl}-2,3-dihydro-1H-imidazol-2-one
2-(4-chloro-2-methylphenoxy)-1-(4-{5-[(1E)-prop-1-en-1-yl]-2-(pyridin-3-yl)pyrimidin-4-yl}piperidin-1-yl)ethan-1-one
3-ethyl-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-{[7-chloro-2-(4-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)furan-2-carboxamide
3-[2-chloro-4-(pyrrolidin-1-ylmethyl)phenoxy]-2,5-dimethylpyrazine
(1S,5R)-3-(3-chloropyridin-2-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,5R)-6-(pyridin-2-ylmethyl)-3-(thiophene-2-sulfonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[2-(methylsulfanyl)ethyl]-4-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
5-[(2-chlorophenyl)methyl]-5-{1-[3-(furan-2-yl)propanoyl]piperidin-4-yl}-3-(2-methoxyethyl)imidazolidine-2,4-dione