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4-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1-(2-methoxyphenyl)piperazin-2-one
methyl (2S,4S)-4-(5-chloro-3-methyl-1H-indole-2-amido)-1-[(3,5-dimethoxyphenyl)methyl]pyrrolidine-2-carboxylate
N-[(3R,4R)-1-[3-(2-fluorophenyl)propanoyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
9-(2-chlorobenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-chloro-4-(4H-1,2,4-triazol-4-yl)benzoyl]-4-(hydroxymethyl)azepan-4-ol
methyl (2S)-2-cyclopropyl-2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)acetate
3-chloro-N-cyclopropyl-4-hydroxy-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
{1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-3-propylpiperidin-3-yl}methanol
methyl 1-[(3R,5S)-5-(azepane-1-carbonyl)-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-methyl-8-{[(4-methylphenyl)methyl]carbamoyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-methyl-N-[(2,3,4-trifluorophenyl)methyl]thian-4-amine
4-{1-hydroxy-2-[(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)amino]ethyl}phenol
3-methoxy-2-{5-[3-(methylsulfanyl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenol
N-benzyl-N-butyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]acetamide
N-{1-[7-(2H-1,3-benzodioxol-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}furan-2-carboxamide
N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[(4-fluorophenyl)methyl]-5-(2-methoxy-4-methylbenzoyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
4-ethyl-3-{1-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]piperidin-3-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
5-(4-tert-butylbenzoyl)-1-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(piperidin-1-ylmethyl)-1-[6-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-ol
1-(4-{3-[({[4-(2-methylpropyl)phenyl]methyl}amino)methyl]pyridin-2-yl}piperazin-1-yl)ethan-1-one
(1R,7S)-3-[(4-fluorophenyl)methyl]-6-(4-methyl-1,4-diazepane-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-(4-ethylpiperazin-1-yl)-3-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)propan-1-one
2-{4-[(3,5-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-1-phenoxypropan-2-ol
methyl (2S,4S)-4-(2-cyclopropylquinoline-4-amido)-1-[(3-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(pyridin-2-ylmethyl)acetamide
5-methoxy-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}furan-2-carboxamide
N-(4-methyl-1,3-thiazol-2-yl)-2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}acetamide
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl})methylamine
N-tert-butyl-8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
1-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}butan-1-one
[(4-ethylphenyl)methyl](methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyridin-2-yl)ethan-1-one
4-{[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-N,N-dimethylpiperidine-1-sulfonamide
2-(2,3-dimethoxyphenyl)-5-methyl-4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-1,3-oxazole
4-(3-methylphenoxy)-1-(pyrrolidine-1-carbonyl)piperidine-4-carboxylic acid
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]ethan-1-one
7-(5-chloropyridin-2-yl)-9-methoxy-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl[2-(morpholin-4-yl)propyl][(2,3,4-trimethoxyphenyl)methyl]amine
(3S,5R)-5-[(6-methylpyridin-3-yl)carbamoyl]-1-(pent-4-enoyl)piperidine-3-carboxylic acid
3-[({[4-(3-fluorophenyl)oxan-4-yl]methyl}amino)methyl]pyrrolidin-3-ol
1-(2,6-dimethylpyridin-4-yl)-4-[3-(methylsulfanyl)butyl]piperazine
2,3-dimethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
4-(quinoxalin-6-ylmethyl)-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide
4-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)phenyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[3-(1H-pyrazol-1-yl)propyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
N,N-dimethyl-2-[2-({3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}methyl)phenoxy]acetamide