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N,N-dimethyl-2-(1,4-oxazepan-4-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-sulfonamide
1-[1-(2-chlorobenzoyl)piperidin-4-yl]-N-cyclopentyl-1H-1,2,3-triazole-4-carboxamide
N-(3-{2-[(dimethylamino)methyl]phenoxy}phenyl)acetamide
methyl 9-(cyclopentyloxy)-3-[(2-methoxynaphthalen-1-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-{[7-(3,5-dimethylbenzoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine-4-carboxamide
N-(cyclopropylmethyl)-N-(oxolan-2-ylmethyl)-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
2-[5-(1-methyl-5-phenyl-1H-pyrrol-2-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-(3-methylphenyl)piperidine
2-(2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-ylmethyl}phenoxy)acetic acid
1-[4-(2-phenoxyethyl)piperazin-1-yl]-2-(thiophen-3-yl)ethan-1-one
1-[(3-fluorophenyl)methyl]-N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-6-oxopiperidine-3-carboxamide
1-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}-2-(naphthalen-2-yloxy)propan-1-one
1-(2-{[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]amino}-4-methylpyrimidin-5-yl)ethan-1-one
1-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}pentane-1,4-dione
4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-[2-(dimethylamino)ethyl]pyrrolidin-2-one
3-{2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{5-[(2S)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
3-benzoyl-1-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidine
N-[2-(diethylamino)ethyl]-2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(1R,9S)-5-amino-12-methyl-3-(1-phenyl-1H-pyrazol-5-yl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-[(4-fluorophenyl)methyl]-1-methyl-5-{[2-(morpholin-4-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2,4-difluorophenyl)-2-(morpholin-4-ylmethyl)piperidine-1-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(2,6-dimethylpyridin-4-yl)pyrrolidin-3-yl]-2-hydroxyacetamide
4-[1-(1,3-thiazol-4-ylmethyl)piperidin-3-yl]benzoic acid
1-butyl-4-(7-methoxy-4-methylquinazolin-2-yl)piperazin-2-one
5-[(2-fluoro-4-methoxyphenyl)methyl]-5-[3-(3-methylpiperidin-1-yl)-3-oxopropyl]pyrrolidin-2-one
1-(benzenesulfonyl)-N-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-amine
2-({[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}(thiophen-3-ylmethyl)amino)butan-1-ol
2-[4-({3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)phenoxy]acetic acid
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetamide
methyl 3-{4-[(4-acetyl-4-phenylpiperidin-1-yl)methyl]-1H-pyrazol-1-yl}propanoate
3-(1-methylpiperidin-3-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
9-(3-hydroxybenzoyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-1-(3-aminopropyl)-6-[2-(cyclohex-1-en-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
2-[3-(propan-2-yl)-5-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)phenyl]-1H-1,2,4-triazol-1-yl]pyridine
6-(4-chlorophenyl)-N-[3-(propan-2-yloxy)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-butyl-8-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
3-{[1-(2-methoxy-2-methylpropanoyl)pyrrolidin-3-yl]methyl}benzoic acid
2-(2H-1,3-benzodioxol-5-yl)-N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
1'-(1,3-benzoxazol-2-yl)-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[3-({4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenyl]ethan-1-one
4-(2-methylpyrrolidine-1-carbonyl)-N-(oxan-4-yl)benzene-1-sulfonamide
N-[(3,4-difluorophenyl)methyl]-3-[1-(quinoxaline-5-carbonyl)piperidin-3-yl]propanamide
2-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methoxypyrazine
3-(4-methoxy-3,5-dimethylbenzoyl)-1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidine
1-[2-(3-methoxypropyl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-amino-6-methyl-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrimidine-4-carboxamide
1-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-2-methyl-1,4-dihydroquinolin-4-one