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2-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-1H-indole
4-[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]-2-methoxypyridine-3-carbonitrile
4-[(1-benzylpiperidin-4-yl)oxy]-3-chloro-N-[2-(dimethylamino)ethyl]benzamide
2-(1H-1,2,4-triazol-1-yl)-3-{[2-(2,4,5-trimethylphenyl)-1H-imidazol-1-yl]methyl}pyridine
(1S,5R)-3-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(morpholin-4-yl)-3-{3-[({2-[4-(propan-2-yloxy)phenyl]ethyl}amino)methyl]phenoxy}propan-2-ol
6-[3-fluoro-5-(trifluoromethyl)phenyl]-N-methylpyridazin-3-amine
N,N-bis(prop-2-en-1-yl)-2-[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]acetamide
3-[2-(dimethylamino)ethyl]-1-[2-(4-methoxyphenyl)ethyl]-8-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2R,3R)-2-methoxy-1'-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
5-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
2-(2,6-difluorophenyl)-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
6-{2-azabicyclo[2.2.1]heptan-2-ylmethyl}-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{5-[(3R)-3-hydroxy-3-phenylpropyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
(1R,5R)-6-(cyclopropylmethyl)-3-[1-(propan-2-yl)-1H-pyrazole-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(4aR,8aS)-1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
3-[2-(3-benzoylpiperidin-1-yl)-2-oxoethyl]-1-cyclopentyl-3-(3-fluorophenyl)pyrrolidine-2,5-dione
6-fluoro-8-(trimethylpyrimidin-4-yl)quinoline
5-(1-{2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-3-(2-methylpropyl)-1,2,4-oxadiazole
2-(2-amino-4,7-dimethyl-1,3-benzothiazol-6-yl)benzamide
(3S,4S)-4-(dimethylamino)-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidin-3-ol
5-ethyl-2,3-dimethyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-(dimethylamino)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
4-[(5-ethylpyridin-2-yl)methyl]-1-(3-methoxyphenyl)piperazin-2-one
[2-(2-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl}-1H-imidazol-1-yl)ethyl]dimethylamine
2-[(5-{[(butan-2-yl)(thiophen-3-ylmethyl)amino]methyl}pyrimidin-2-yl)amino]acetic acid
(4aR,7aS)-1-cyclopropanecarbonyl-4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(dimethylamino)-N-methyl-N-[1-(1-{2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetyl}piperidin-4-yl)-2-phenylethyl]acetamide
1-(4-chloro-1H-pyrazole-3-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-[4-(propan-2-yl)morpholin-2-yl]acetamide
2-(6-methoxynaphthalen-2-yl)-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}morpholine
N,6-dimethyl-N-(oxan-4-ylmethyl)-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
6-(2-aminoethyl)-N,2-dimethyl-N-(thiophen-3-ylmethyl)pyrimidin-4-amine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(phenylsulfanyl)acetamide
2-[(2,3-dihydro-1,4-benzodioxin-6-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-(3-cyclopropyl-5-{6-methylimidazo[2,1-b][1,3]thiazol-3-yl}-1H-1,2,4-triazol-1-yl)-3-methylpyridine
3-(4-fluorophenoxymethyl)-1-(1,2-oxazole-3-carbonyl)piperidine
N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-(oxolan-3-yl)acetamide
1-[2-(2-ethoxyethoxy)benzoyl]-3-(1H-imidazol-2-yl)piperidine
2-(1-ethyl-1H-pyrazol-4-yl)-5,7-dimethyl-4-(2-methylpiperidine-1-carbonyl)quinoline
1-[1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperidin-3-yl]pyrrolidin-2-one
4-[1-(2-hydroxybutyl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl]-1-methyl-1,2-dihydroquinolin-2-one
2-(4-{[1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}piperazin-1-yl)pyrimidine
2-methyl-N-[(3-methyl-1H-pyrazol-5-yl)methyl]-6-(propan-2-yl)pyrimidin-4-amine
1-[4-(4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}piperidin-1-yl)piperidin-1-yl]ethan-1-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[2-(pyridin-2-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{4-methyl-3-oxo-1-oxa-4,9-diazaspiro[5.5]undecan-9-yl}-2-oxo-N-phenylacetamide
[(5-chloro-1-benzothiophen-3-yl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
1-(2-methoxy-4-{[(3-phenylpropyl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
6-methoxy-N,3-dimethyl-N-(quinolin-5-ylmethyl)-1-benzofuran-2-carboxamide