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N-[(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-3-(pyridin-3-yl)propanamide
N-(adamantan-2-yl)-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
N-({3-[4-(methylsulfamoyl)phenyl]phenyl}methyl)propanamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]amino}pyrrolidine-2-carboxamide
methyl 3-(3-methylbutyl)-2-oxo-1-(1,3-thiazol-5-ylmethyl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
2-({5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}methyl)pyridine
{5-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-2-yl}methanol
1-[2-(dimethylamino)ethyl]-3-[(4-fluorophenyl)methyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
2-[3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-2,5-dioxopyrrolidin-3-yl]-N-[(4-fluorophenyl)methyl]-N-methylacetamide
1,3,7-trimethyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1H-indole-2-carboxamide
2-(morpholin-3-yl)-N,N-bis(pyridin-3-ylmethyl)acetamide
9-(1-methyl-1H-indole-3-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
methyl({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]amine
4-chloro-1,3-dimethyl-N-[(3-propoxyphenyl)methyl]-1H-pyrazole-5-carboxamide
1-(1H-imidazol-4-ylmethyl)-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
2-(3-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}-1H-indol-1-yl)-N-(propan-2-yl)acetamide
5-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}-2-methylphenol
1-(furan-3-ylmethyl)-3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
3-(piperidine-1-carbonyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]benzene-1-sulfonamide
2-(phenylsulfanyl)-N-[1-({[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]acetamide
2-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
5-methyl-4-{5-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}-3-phenyl-1,2-oxazole
N-(5-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-2-phenoxyacetamide
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(furan-2-carbonyl)-1,4-diazepane
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}imidazo[1,2-a]pyridine-3-carboxamide
8-(1H-1,2,3-benzotriazole-5-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2,3-dihydro-1H-inden-4-yl)-4-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)benzamide
N-ethyl-2-methyl-N-[2-(4-methylbenzenesulfonyl)ethyl]-1,3-thiazole-4-carboxamide
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[(2-methylnaphthalen-1-yl)methyl]pyrrolidin-3-yl]methanol
1-methyl-6-(2-phenylethyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-methoxy-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-cyclohexyl-6-(pyridin-2-ylmethoxy)-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepan-2-one
2-(4-fluorophenoxy)-1-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]benzamide
(2S,4R)-4-amino-1-[3-(3,4-dimethoxyphenyl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}-1,4-diazepane-1-carbaldehyde
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-[(3-methylthiophen-2-yl)methyl]propanamide
2-amino-4-(dimethyl-1,2-oxazol-4-yl)-6-(2-fluoro-4-methoxyphenyl)pyridine-3-carbonitrile
(1S,5R)-6-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
ethyl 4-benzyl-1-(thiophene-3-sulfonyl)piperidine-4-carboxylate
2-[(phenylsulfanyl)methyl]-6-(piperidin-3-yl)-3,4-dihydropyrimidin-4-one
1-(adamantane-1-carbonyl)-N-(4-fluorophenyl)piperidin-3-amine
N-[(2R,3R)-1'-[(3-acetylphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
3-(4-methoxyphenyl)-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-5-carboxamide
3-(oxolan-3-yl)-5-[(2-phenyl-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-[(3-methoxyphenyl)sulfanyl]ethan-1-one
N-[2-(2-methylpropanesulfonyl)ethyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
3-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyridazine
N-{2-[(2-methyl-4-phenylpyrimidin-5-yl)formamido]ethyl}pyridine-3-carboxamide