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N-[2-(3-hydroxypiperidin-1-yl)ethyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
1-(2-methoxy-5-phenylphenyl)-3-(2-methoxybutyl)urea
6-(hydroxymethyl)-N-(1-oxo-2,3-dihydro-1H-inden-5-yl)-1,4-oxazepane-4-carboxamide
3-(2-chlorophenyl)-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidine
1-methyl-4-[3-(2-methyl-1,3-thiazol-4-yl)-5-[1-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazol-1-yl]piperidine
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(1-phenylcyclopropyl)benzamide
N-methyl-5-(4-methylpiperidin-1-yl)-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopentyl-2-(morpholin-2-yl)acetamide
2-(3-{[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]methyl}phenyl)-5-fluoro-6-methyl-3,4-dihydropyrimidin-4-one
4-[3-(2-fluorophenoxy)azetidine-1-carbonyl]-1-(pyridin-4-ylmethyl)pyrrolidin-2-one
5-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-1-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]ethan-1-one
methyl 2-[(butan-2-yl)sulfamoyl]-6-(2,4-difluorobenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-cyclohexyl-5-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1,2,4-oxadiazole
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}acetamide
[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl](methyl)[(1-methylpyrrolidin-2-yl)methyl]amine
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)methylamine
N,N-bis(1,3-oxazol-4-ylmethyl)-4-(2-oxopyrrolidin-1-yl)benzamide
({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)[2-(pyrrolidine-1-sulfonyl)ethyl]amine
N-({7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzenesulfonamide
8-[(2-hydroxy-4-methoxyphenyl)methyl]-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-(4,6-dimethylpyridine-3-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
4-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}pyrimidin-2-amine
1-(2-methoxyphenyl)-3-{1-[1-(1-methylpiperidine-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-[2-(dimethylamino)ethyl]-2-(3-fluorophenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
5-methoxy-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]furan-2-carboxamide
methyl 2-[4-(benzyloxy)piperidine-1-carbonyl]piperidine-1-carboxylate
1-({5-[1-(methoxymethyl)cyclobutyl]-1,2,4-oxadiazol-3-yl}methyl)-4-methylpiperazine
N-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)acetamide
1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2-methoxy-N-[3-methyl-1-(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)butyl]acetamide
4-{5-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2-methoxyphenol
5-(2,4-difluorophenoxymethyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
N-(1-{7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)propanamide
N-[(3R,4S)-4-cyclopropyl-1-[(4-methoxy-3-methylphenyl)methyl]pyrrolidin-3-yl]-2-hydroxyacetamide
4-(dimethyl-1,3-thiazole-5-carbonyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
2-(4-chlorophenyl)-N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
7-methyl-3-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-4-(pyridin-3-yl)piperidin-4-ol
(2E)-N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]-3-(thiophen-2-yl)prop-2-enamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]propanamide
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
6-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyrazine-2-carboxamide
N-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
1-(2-methoxyphenyl)-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}-1H-pyrazole-4-carboxamide
1-(4-ethylbenzenesulfonyl)-3-(3-methylthiophene-2-carbonyl)piperidine
N-(2-{1-[(3-chloro-4,5-dimethoxyphenyl)methyl]piperidin-2-yl}ethyl)acetamide
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-cyclopropyl-3-[1-(propan-2-yl)-5-[(propan-2-yl)sulfamoyl]-1H-1,3-benzodiazol-2-yl]propanamide