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4-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-1-ethyl-1H-pyrrole-2-carbonitrile
ethyl 1-(2-methoxyethyl)-5-(quinoxalin-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[2-(dimethylamino)ethyl]-3-(3-fluorophenyl)-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]pyrrolidine-2,5-dione
1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxylic acid
(1-{4-[(diethylamino)methyl]-5-ethylfuran-2-carbonyl}piperidin-2-yl)methanamine
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
methyl 3-(naphthalen-2-ylmethyl)-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)propan-1-ol
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-3-(1-methyl-1H-pyrazol-4-yl)propanamide
4-(5-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
1-[2-(piperidin-1-yl)acetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-chloro-4-{[1-(2-cyclopentylacetyl)piperidin-4-yl]oxy}-N-[2-(dimethylamino)ethyl]benzamide
6-(4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine-2-carbonitrile
5-methyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2S,4S)-N-ethyl-4-(5-methoxyfuran-2-amido)-1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]pyrrolidine-2-carboxamide
N-benzyl-N-(oxolan-2-ylmethyl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(3-methylthiophen-2-yl)ethyl]acetamide
2-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)-3,5-dimethyl-1,4-dihydropyridin-4-one
(3aR,6aR)-2-methanesulfonyl-5-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(4-{[3-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
2-{1-methyl-10-oxo-4-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
1-(1-{2-[(4-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-4-carbonyl)-N,N-diethylpiperidine-3-carboxamide
1-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
(1S,5R)-6-methyl-3-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{[2-(6-hydroxy-1,4-oxazepane-4-carbonyl)phenyl]sulfanyl}-1-phenylethan-1-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
2-[3-(pyrimidin-4-yl)piperidine-1-carbonyl]pyridin-3-ol
4-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
2-amino-4-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]-3-phenylpropanamide
1-(2-fluoro-5-methylphenyl)-3-[3-(1H-1,2,4-triazol-1-yl)propyl]urea
1-cyclohexyl-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
2-(2,5-dimethoxyphenyl)-N-(3-methoxypropyl)-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}acetamide
(1H-indol-3-ylmethyl)[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
N-[2-(diethylamino)ethyl]-N-ethyl-1-[2-(3-fluorophenyl)ethyl]-6-oxopiperidine-3-carboxamide
N-methyl-2-(methylamino)-N-{[3-(methylsulfanyl)phenyl]methyl}pyridine-4-carboxamide
1-(3-{[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenyl)ethan-1-one
6-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-[(3R,4S)-3-(1-methyl-1H-pyrazole-4-amido)-4-(propan-2-yl)pyrrolidin-1-yl]butanoic acid
N-(1-{4-[4-(5-chloro-2-methylphenyl)piperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)furan-3-carboxamide
[(5-chlorothiophen-2-yl)methyl]({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]benzamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-[4-(2-methylquinolin-6-yl)-1H-pyrazol-1-yl]acetamide
N-(3-chloro-4-methoxyphenyl)-3-(5-fluoro-2-methoxybenzoyl)piperidine-1-carboxamide
N-[3-(5-methyl-4-{[4-(thiophen-2-yl)butanamido]methyl}-1,3-oxazol-2-yl)phenyl]pyridine-4-carboxamide
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-1-{1-oxa-7-azaspiro[3.5]nonan-7-yl}butan-1-one
(3S,4R)-1-(2-cyclopentylacetyl)-4-(2,3-dimethoxyphenyl)pyrrolidine-3-carboxylic acid
4-(1H-indol-3-ylmethyl)-1-(3-methoxyphenyl)-6-methylpiperazin-2-one
(2-methoxyethyl)[(1-methyl-1H-imidazol-2-yl)methyl][(4-methylphenyl)methyl]amine