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1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
N-({7-[2-(2-methoxyphenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-5-carboxamide
[(1-{1-[(2E)-hex-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]urea
(4aR,7aS)-1-(2-methylpropanoyl)-4-[3-(thiophen-3-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(3-methylpyridin-2-yl)methyl]-4-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
N-[(1-cycloheptylpyrrolidin-3-yl)methyl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
4-(2-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}ethyl)benzene-1-sulfonamide
2-(dimethylamino)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(2-methylphenyl)-N-(2-methylpropyl)acetamide
2-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-methoxypyrazine
[(3R,4R)-1-[1-(3,4-difluorophenyl)piperidin-4-yl]-4-{[ethyl(methyl)amino]methyl}pyrrolidin-3-yl]methanol
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-3-(4-methylpiperazine-1-carbonyl)benzene-1-sulfonamide
4-{2-[2-(thiophen-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}benzene-1-sulfonamide
4-({5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}amino)butan-1-ol
6-methoxy-3-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)-1,2-dihydroquinolin-2-one
N-cyclopentyl-2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2,3-dihydro-1H-indene-2-carboxamide
7-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]-2,3-dimethyl-1H-indole
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(1,2-oxazol-5-ylmethyl)amino]methyl}piperidin-2-one
6-methoxy-N-(oxan-4-yl)-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}cycloheptanamine
2-{2-[4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,2-benzothiazol-3-one
1-[cyclohexyl(methyl)amino]-3-{3-[(4-methylpiperazin-1-yl)methyl]phenoxy}propan-2-ol
1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidine-1-carbonyl)cyclopropane-1-carboxamide
3-(1-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}piperidin-2-yl)pyridine
8-methoxy-5-(6-methoxypyridazin-3-yl)-2-methylquinoline
{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
1-(2-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-oxoethyl)-5,5-dimethylimidazolidine-2,4-dione
methyl 4-({[2-(5-oxo-1-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}pyrrolidin-2-yl)ethyl]amino}methyl)benzoate
1-[1-(2-methylpyridin-4-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]cyclopropane-1-carboxamide
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-[2-(prop-2-en-1-yloxy)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2,6-dimethyl-N,N-bis(1,3-oxazol-4-ylmethyl)quinoline-3-carboxamide
2-(4-fluorophenoxymethyl)-N-[2-(piperidin-1-yl)ethyl]-1,3-oxazole-4-carboxamide
9-(1-ethyl-1H-pyrazole-5-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-methyl-1-{2-[4-(2-phenyl-1,3-oxazol-4-yl)-1H-1,2,3-triazol-1-yl]ethyl}piperidine
3-(2-chlorophenyl)-1-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}propan-1-one
(3S,7S)-5-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2,2-dimethylpropyl)-3-hydroxy-3-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)piperidin-2-one
2-(adamantan-1-yl)-N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]acetamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propan-1-one
2-{4-[(1-methyl-1H-imidazol-5-yl)methyl]piperazin-1-yl}pyrazine
4-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}thiomorpholine
3-[4-(4-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]-N,N-dimethylpropane-1-sulfonamide
{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[1-(pyrazin-2-yl)propan-2-yl]amine
N-[(3S,5S)-5-[(1H-imidazol-2-ylmethyl)(methyl)carbamoyl]-1-methylpyrrolidin-3-yl]morpholine-4-carboxamide
3-[3-cyclopropyl-5-(2-methylphenyl)-1H-1,2,4-triazol-1-yl]-4-fluorobenzene-1-sulfonamide
ethyl 1-{[(4-chloro-1-methyl-1H-indazol-3-yl)carbamoyl]methyl}-1H-imidazole-2-carboxylate
(4aR,6R,8aS)-2-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinoline
3-(4-fluoro-3-methylphenyl)-6-(3-phenylpropanoyl)-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one