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N-(1H-indazol-7-yl)-3-(4-methoxyphenoxymethyl)piperidine-1-carboxamide
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(methylsulfanyl)propanamide
2-{[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]methyl}benzonitrile
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-(diphenylmethyl)acetamide
3-{[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-2,4-dichlorophenol
4-(2-methylpyrrolidine-1-carbonyl)-N-(pyridin-4-ylmethyl)benzene-1-sulfonamide
1-cyclohexyl-N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
5-[2-(methylsulfanyl)phenoxymethyl]-N-{2-[3-(trifluoromethyl)phenyl]ethyl}-1,2-oxazole-3-carboxamide
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-[3-(methylsulfanyl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl (2S,4R)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]-1-[(4-ethylphenyl)methyl]pyrrolidine-2-carboxylate
1-ethyl-5-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H,4H-pyrazolo[3,4-d]imidazole
4-(cyclohexylmethyl)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1,4-diazepan-5-one
N-[2-(4-chlorophenyl)-2-hydroxyethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]acetamide
N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
7-fluoro-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
8-[2-(2,4-dimethylphenoxy)ethyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
2-[(adamantan-1-ylmethyl)({[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl})amino]ethan-1-ol
2,2-diethyl-4-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]morpholine
(3aR,6aR)-2-acetyl-5-{[4-(methylsulfamoyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3S,4S)-4-cyclopropyl-1-(4-methoxypyrimidin-2-yl)pyrrolidine-3-carboxylic acid
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanamide
4-phenyl-N-({1-[3-(1H-pyrazol-4-yl)propanoyl]piperidin-3-yl}methyl)benzamide
N-(2-{[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}quinolin-6-yl)acetamide
({2-[(3-fluorophenyl)methoxy]-6-methylquinolin-3-yl}methyl)[(3-methyloxetan-3-yl)methyl]amine
1-(2-chloroprop-2-en-1-yl)-3-({[(4-fluorophenyl)methyl]amino}methyl)-6,7-dimethoxy-1,2-dihydroquinolin-2-one
methyl (2S)-1-{2-[2,5-dioxo-3-phenyl-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]acetyl}pyrrolidine-2-carboxylate
9-({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)-6-oxa-9-azaspiro[4.5]decane
8-(propane-2-sulfonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-cyclopentyl-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-5-oxopyrrolidine-3-carboxamide
6-chloro-N,N-dimethyl-3-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-2-methyl-1-benzofuran-5-carboxamide
3-({2-[2-(trifluoromethyl)phenyl]-1H-imidazol-1-yl}methyl)pyridine
2-methyl-4-{4-[4-(pyridin-4-yl)piperazine-1-carbonyl]phenyl}butan-2-ol
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
6-(4-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}piperazin-1-yl)pyridine-2-carbonitrile
ethyl 4-[7-(1-benzothiophen-3-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidine-1-carboxylate
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
2-cyano-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)benzamide
3-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]-5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
N-ethyl-1-(6-methoxy-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
N-benzyl-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(cyclohex-1-en-1-ylmethyl)-2-{4-[(4-methoxy-2,3-dimethylphenyl)methyl]morpholin-3-yl}acetamide
3-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-4,5,6,7-tetrahydro-1,2-benzoxazole
N-[(3-fluorophenyl)methyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
N-[1-cyclopentyl-7-(3-propanoylpiperidine-1-carbonyl)-1H-1,3-benzodiazol-5-yl]benzamide
1-[(2,3-dimethoxyphenyl)methyl]-4-[(3-fluorophenyl)methyl]piperazine