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N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
8-(2H-1,3-benzodioxol-5-ylmethyl)-1-methyl-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-6-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}-1H-indole
(3S,4S)-4-(naphthalen-2-yl)-1-(piperidin-4-ylmethyl)piperidin-3-ol
N-ethyl-2-{4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]morpholin-3-yl}acetamide
4-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-1-ethylpyrrolidin-2-one
3-propyl-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-4-(oxolane-2-carbonyl)-1,4-diazepane
3-{2-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
2-ethoxy-5-[2-(phenoxymethyl)pyrimidin-4-yl]benzoic acid
(3R,4R)-1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-(hydroxymethyl)piperidin-3-ol
(5S,9aS,9bS)-5-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-({3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}methyl)imidazolidine-2,4-dione
1,5-dimethyl-4-({1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-1H-pyrazole
2-methyl-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-1-benzofuran-5-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1,1-dioxo-1λ6-thiane-4-carboxamide
4-benzyl-1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-2-one
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl){[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
N-[(3S,4R)-1-(5-phenoxyfuran-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
6-(2-fluorophenyl)-N-[(3S)-2-oxoazepan-3-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-ethyl-4-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
3-(1-{[1-(9H-purin-6-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-1-ol
5-(2-fluoro-5-methoxyphenyl)thiophene-2-carboxamide
5-(3-methylbut-2-en-1-yl)-1'-(pyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(piperidin-1-ylmethyl)-4-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-1,4-oxazepane
2-methyl-5-{2-oxo-2-[2-(trifluoromethyl)morpholin-4-yl]ethyl}-3,4-dihydropyrimidin-4-one
1-(thiophen-3-ylmethyl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazine
1-cyclobutanecarbonyl-N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]piperidine-4-carboxamide
9-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]-3-azaspiro[5.5]undecane
6-(3-phenylpropyl)-N-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
2-(4-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
5-methyl-N-{[4-(methylsulfanyl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(2-chlorophenyl)ethyl]-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
6-{[3-(4-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-{1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carbonyl}-N,N-diethylpyrrolidin-3-amine
1-[(4-fluorophenyl)methyl]-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N-(2-methoxyethyl)-1-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
(2S)-2-[(4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methylthieno[2,3-d]pyrimidin-6-yl)formamido]-4-methylpentanamide
N-[3-(4-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)propyl]cyclopropanecarboxamide
4,6-dimethyl-N-{2-[1-(2-methylpropyl)piperidin-3-yl]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
2-{3,9-diazaspiro[5.5]undecan-3-yl}propane-1,3-diol
2-{3-[3-(3,6-dimethylpyrazin-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
5-[(2-chlorophenyl)methyl]-3-(pentan-3-yl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
N-[(3-ethoxyphenyl)methyl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
(2R,3S,6R)-5-(furan-2-ylmethyl)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[3-(cyclohexylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
N-cyclopropyl-N-(1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-(2,2-diphenylethyl)-N-(furan-3-ylmethyl)-N-methylpyrrolidine-2-carboxamide
3-({methyl[4-(morpholin-4-yl)butyl]amino}methyl)phenol