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2-(4-methoxyphenyl)-5-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}pyrimidine
4-cyano-N-cyclohexyl-N-[2-(1H-indol-3-yl)ethyl]-1H-pyrrole-2-carboxamide
(4aS,7aR)-1-[(2-methoxyphenyl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-N-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}oxolan-3-amine
1-{[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-4-(4-ethyl-1H-pyrazol-5-yl)piperidine
5,6-dimethyl-3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}benzamide
(2S,4S)-N-[(4-methylphenyl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
1-cyclopentyl-N-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
5-(methoxymethyl)-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)thiophene-2-carboxamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-N-(pyridin-3-ylmethyl)-4-(1H-1,2,4-triazol-1-yl)butanamide
4-[(5-methylfuran-2-yl)methyl]-7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[(4-chlorophenyl)methyl]-5-(1,2-oxazolidine-2-carbonyl)-1,3-benzoxazole
1-(2-methoxyphenyl)-4-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)piperazine
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(3-methoxyphenyl)acetamide
N-benzyl-4-[(1-methoxybutan-2-yl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-3-(2-fluorophenyl)-N-(pyridin-3-ylmethyl)propanamide
2-cyclobutyl-N-[(2,5-dimethoxyphenyl)methyl]-1-methyl-7-(oxolane-2-amido)-1H-1,3-benzodiazole-5-carboxamide
5-cyclobutanecarbonyl-1'-(1H-pyrazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(1-{7-[(4-ethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-5-(methoxymethyl)furan-2-carboxamide
2-(2,8-dimethylquinoline-3-carbonyl)-8-methyl-2,8-diazaspiro[4.5]decane
2-(1H-imidazol-2-yl)-N-methyl-N-[1-(pyridin-3-yl)propyl]benzamide
4-(4-chlorophenoxy)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-5-(oxolan-2-yl)thiophene-2-carboxamide
1-ethyl-N-(1H-indol-3-yl)-1H-pyrazole-4-carboxamide
2-{4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
1-[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]-4-phenylpiperidin-4-ol
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)benzamide
methyl 2-(diethylsulfamoyl)-6-(3-methylpentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-benzyl-4-[3-(5-methylfuran-2-yl)benzoyl]piperazin-2-one
2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-1,3-benzoxazole
3-(1,2-oxazinan-2-yl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]propanamide
methyl 8-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-[3-(pyridin-2-yl)propyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-{2-oxo-2-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrol-1-yl]ethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-{1-[(4-fluorophenyl)methyl]-4-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
1-methyl-4-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1,4-diazepane
1-(3-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}phenyl)ethan-1-one
({5-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-1,3,4-oxadiazol-2-yl}methyl)dimethylamine
1-[(3-methylphenyl)methyl]-4-(thiophene-3-carbonyl)piperazin-2-one
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(1-propylpiperidin-4-yl)benzamide
2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-{3-[(methylsulfanyl)methyl]piperidin-1-yl}ethan-1-one
(2S)-2-amino-N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]hexanamide
3-(1-ethyl-1H-pyrazol-5-yl)-1-{1-phenyl-3,6-diazatricyclo[4.3.1.13,8]undecan-9-yl}urea
2-{4-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-fluoro-5-methylphenyl)methyl]piperidine
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1,4-diazepan-1-yl]-6-ethoxy-4-methylquinazoline
N-cyclohexyl-2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propanamide
2-cyclobutyl-1-methyl-7-(oxolane-2-amido)-N-(pyridin-4-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
(5-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}furan-2-yl)methanol