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5-fluoro-3-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-4-yl)-1,2-benzoxazole
2-{4-[(4-fluorophenyl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
4-[({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)carbamoyl]pyridin-1-ium-1-olate
8-(3-chloropyridin-2-yl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-decahydro-1,6-naphthyridin-2-one
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-[2-(1H-indol-1-yl)ethyl]-N-methylacetamide
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-2,3-dimethyl-N-(pyridin-3-ylmethyl)-1H-indole-7-carboxamide
2-(morpholin-2-yl)-N-{[4-(trifluoromethoxy)phenyl]methyl}acetamide
2-[(5-ethyl-2-methylpyrimidin-4-yl)amino]-N-(5-fluoro-2-methylphenyl)propanamide
N-[1-(7-{[4-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-3-phenylpropanamide
methyl[(4-methyl-1H-imidazol-2-yl)methyl]{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(2S)-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-2-carboxamide
2-methyl-3-(morpholin-4-yl)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]propan-1-one
3-({5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)propan-1-ol
5-(4-methanesulfonylphenyl)-4-phenyl-1H-imidazole
3-[(3-fluorophenyl)methyl]-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)furan-2-carboxamide
4-(4-chlorophenyl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]butanamide
2-amino-4-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
6-{methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
2-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-7-methyl-2,7-diazaspiro[4.4]nonane
N-[2-(cyclohex-1-en-1-yl)ethyl]-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
[7-(3,5-difluoro-4-methoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
4-phenyl-1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,2,3,6-tetrahydropyridine
5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-4-propylpyrimidine
2-(dimethylamino)-N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]pyridine-3-carboxamide
4-[4-(2,4-dimethylphenyl)-1H-imidazol-2-yl]-1-(2-methylpropyl)pyrrolidin-2-one
3-(4-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)propanamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-[(1-benzylpiperidin-4-yl)amino]-1-[(4-chlorophenyl)methyl]pyrrolidine-2-carboxamide
1-[4-({4-[4-(2-fluorophenyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
2-[4-(1-benzofuran-2-ylmethyl)-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl]ethan-1-ol
2-methoxy-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}quinoline
1-[(1-methyl-1H-imidazol-5-yl)methyl]-3-(3-{pyrazolo[1,5-a]pyrimidin-3-yl}phenyl)-1H-pyrazole
2-(2-methyl-1,3-thiazol-4-yl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-[2-(2,5-dimethylphenyl)acetyl]-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(3S,4S)-1-{5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-methylpiperidine-3,4-diol
3-chloro-4-{[1-(2,2-diethylcyclopropanecarbonyl)piperidin-4-yl]oxy}-N-[2-(dimethylamino)ethyl]benzamide
1-(cyclohexylmethyl)-N-[(5-fluoro-2-methylphenyl)methyl]-6-oxopiperidine-3-carboxamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-cyclopropyl-5-oxopyrrolidine-3-carboxamide
N-[(2-ethoxypyridin-3-yl)methyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-{2-[4-(4-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-1-(3-methoxypropyl)-3-phenylpyrrolidine-2,5-dione
4-(2-methylphenyl)-3-(3,4,5-trimethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[5-(dimethylsulfamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-[2-(5-methylthiophen-2-yl)ethyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
[1-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)piperidin-4-yl]methanol
3-{1-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-pyrazol-4-yl}benzoic acid
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-5-[(isoquinolin-5-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-ethyl-2-(2-oxo-1,2-dihydroquinoxalin-1-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide