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3,5-dimethoxy-2-[(3-methoxypyrrolidin-1-yl)methyl]benzoic acid
4-[3-(propan-2-yloxy)propyl]-11-{[(3,4,5-trifluorophenyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
methyl 3-(oxolane-2-amido)-1-(2-phenylethyl)-5-(propylamino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
8-[(2-methoxynaphthalen-1-yl)methyl]-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-5-methyl-6-(4-methylphenyl)pyridine-3-carbonitrile
1-methyl-3-({[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}sulfanyl)-1H-indole
2-({4-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(2-fluorophenyl)acetamide
1-[(diethylcarbamoyl)methyl]-N-[(2,6-difluoro-3-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-{[4-(2-methyl-6-propylpyrimidin-4-yl)piperazin-1-yl]methyl}-1H-1,3-benzodiazole
6-[2-(3-fluorophenyl)azepane-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[4-methyl-7-(methylsulfanyl)quinolin-2-yl]-1,4-diazepan-5-one
N,4-dimethyl-2-(propan-2-yl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-thiazole-5-carboxamide
1-(4-fluorophenyl)-6,6-dimethyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
(2H-1,3-benzodioxol-4-ylmethyl)(furan-2-ylmethyl)(prop-2-en-1-yl)amine
N-[(1R,2R)-1-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)-2,3-dihydro-1H-inden-2-yl]acetamide
2-methyl-6-{1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperidin-4-yl}pyrimidin-4-ol
N-(1-{7-[(4-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
6-cyano-N-ethyl-N-(oxolan-2-ylmethyl)pyridine-3-carboxamide
4-cyano-1-methyl-N-(morpholin-2-ylmethyl)-1H-pyrrole-2-carboxamide
N-(1-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
4-[2-methoxy-5-(propan-2-yl)phenyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
ethyl 4-({4-[(1-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperidin-3-yl)methoxy]phenyl}methyl)piperazine-1-carboxylate
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
N-{[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)pyrrolidin-3-yl]methyl}-2-methoxyacetamide
methyl 2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}hexanoate
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-cyclopentanecarbonyl-N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]piperidine-4-carboxamide
3-(furan-2-yl)-1-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidin-1-yl}propan-1-one
N-[(3-methyl-7-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(thiophen-3-yl)acetamide
3-methoxy-2,2-dimethyl-N-[1-(3-methylphenyl)cyclopropyl]propanamide
(4aS,8aR)-6-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
8-fluoro-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methylquinoline-2-carboxamide
5-acetyl-N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)thiophene-2-carboxamide
6-[(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-(4-methanesulfonylphenyl)ethan-1-one
N-[(5-methylpyrazin-2-yl)methyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
2-cyclopentyl-9-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-{1-[(4-fluorophenyl)methyl]-4-{6-[(propan-2-yl)amino]pyrimidin-4-yl}piperazin-2-yl}ethan-1-ol
3-(2,3-dimethoxyphenyl)-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
2-oxo-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-phenylpyrrolidine-3-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
1-(furan-2-ylmethyl)-1-[2-(morpholin-4-yl)ethyl]-3-(quinolin-7-yl)urea
3-methyl-2-(3-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine
1-(4-chloro-2-ethylphenyl)-3-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}urea
1-{[2-(2-hydroxyethoxy)phenyl]methyl}-4-(2-methylquinolin-6-yl)piperidin-4-ol
6-amino-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}hexan-1-one
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-2-hydroxypyridine-3-carboxamide
ethyl 1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate