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N-[(3R,4R)-1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
2-[4-(1H-imidazol-2-yl)piperidin-1-yl]quinoxaline
3-(3-fluorophenyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-4-carboxamide
9-(2-methoxy-6-methylbenzoyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methanesulfonyl-4-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
2-{[1-(diphenylmethyl)-1H-1,2,3-triazol-4-yl]formamido}acetamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
N,N-dimethyl-5-{[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]methyl}-1,3-thiazol-2-amine
2-methyl-4-(3-{4-[(pyrimidin-2-yl)amino]piperidine-1-carbonyl}phenyl)but-3-yn-2-ol
1-(2,6-dimethylpyridin-4-yl)-4-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperazine
3,4-difluoro-N-({4-[4-(2-methoxyphenyl)piperazin-1-yl]quinazolin-2-yl}methyl)benzamide
1-[4-(5-aminopyridin-2-yl)phenyl]-3-butylurea
[(3S,4S)-4-(hydroxymethyl)-1-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidin-3-yl]methanol
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[4-(2-ethylpiperidine-1-carbonyl)-5-methyl-1H-pyrazol-1-yl]-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
N-({8-[(3,5-dimethylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)furan-2-carboxamide
2-ethoxy-5-{2-[(pyridin-2-ylmethyl)amino]pyrimidin-4-yl}benzoic acid
N-[2-(pyridin-3-yloxy)propyl]-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
1-(4,6-dimethylquinazolin-2-yl)-N-(2-phenylpropyl)piperidine-4-carboxamide
N-methyl-2-oxo-N-(quinolin-2-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-2-methyl-N-(pyridin-3-ylmethyl)aniline
4-{[6-(3-methyl-3-phenylpiperidin-1-yl)pyridin-3-yl]methyl}morpholine
N-(but-2-yn-1-yl)-N-(furan-2-ylmethyl)-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-4-{1-[(2,3,6-trifluorophenyl)methyl]piperidin-3-yl}pyrimidine
5-ethyl-1'-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-methyl-N-(1-{1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-4-yl}-2-(2-methylphenyl)ethyl)-2-(1H-pyrazol-1-yl)acetamide
N-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-N-methyloxan-4-amine
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-[2-(3-methoxyphenyl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N3-[2-(3-chlorophenyl)ethyl]-1-(2-methoxyethyl)-4-oxo-N5-(2,2,2-trifluoroethyl)-1,4-dihydropyridine-3,5-dicarboxamide
ethyl 2-({methyl[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]amino}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate
5-{1-[(2-chloro-4,5-dimethoxyphenyl)methyl]piperidin-4-yl}-3-[(4-fluorophenyl)methyl]-5-methylimidazolidine-2,4-dione
2,4,6-trimethyl-3-[3-(1H-pyrazol-3-yl)phenyl]aniline
2-tert-butyl-5-[4-(2-phenylethyl)piperazine-1-carbonyl]pyrimidin-4-ol
2-{1-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-{[4-(methylsulfanyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{1-[1-(2-hydroxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-phenylmethanesulfonamide
methyl 3-({2-[(4-methoxyphenyl)methyl]-1,3-benzoxazol-6-yl}formamido)propanoate
5-chloro-2-fluoro-N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-methyl-3-[methyl({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl})amino]propanamide
3-chloro-4-fluoro-N-[1-(pyrazin-2-yl)propan-2-yl]-1-benzothiophene-2-carboxamide
3-butyl-1-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}urea
({4-[(dimethylamino)methyl]phenyl}methyl)(methyl){[5-(oxan-2-yl)furan-2-yl]methyl}amine
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)butan-1-one
6-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]pyridine-2-carbonitrile
1-[1-(5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
6-cyclopropyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}pyrimidin-4-amine
3-[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-(pyridin-3-yl)propanamide
N-(2-{[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]methyl}quinolin-5-yl)acetamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[1-(methylsulfanyl)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione