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1-cycloheptyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
(3S,4R)-N,N-dimethyl-4-(propan-2-yl)-1-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}pyrrolidin-3-amine
1-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyphenoxy)piperidine
3-(dimethyl-1,2-oxazol-4-yl)-1-{7-[(4-phenylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}propan-1-one
4-[(3-fluorophenyl)methyl]-3-{2-[4-(2-methylphenyl)piperazin-1-yl]-2-oxoethyl}piperazin-2-one
[4-(azepan-1-yl)butyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
(3S,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
(2S)-2-amino-3-(1H-imidazol-4-yl)-N-methyl-N-[(4-phenoxyphenyl)methyl]propanamide
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-1H-imidazole-5-carboxamide
3-[1-(2-methoxyphenyl)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-methoxy-3-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridine
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
4-{4-[(dimethylamino)methyl]thiophen-2-yl}-3-methyl-1-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
methyl 6-[(4-ethylphenyl)methyl]-2-[(oxolan-2-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-ethyl-4-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazin-2-one
N-(4-methoxy-2-methylphenyl)-3-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]propanamide
4-[1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl]pyridine
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
5-{[4-(2-methanesulfonylethyl)piperazin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
5-chloro-3-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-4,6-dimethyl-1,2-dihydropyridin-2-one
(3R,4R)-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]imidazo[1,2-a]pyridine-6-carboxamide
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
(1H-imidazol-2-ylmethyl)({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)amine
4-[2-(5-fluoro-2-methylphenyl)pyridine-4-carbonyl]morpholine
2-{5-[2-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]acetamide
N-(2-methoxyethyl)-1-(3-methylbutyl)-4-oxo-5-(4-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
4-(2-{1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]piperidin-2-yl}ethyl)morpholine
3-(azetidine-1-sulfonyl)-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-(thiophen-3-yl)acetamide
1-ethyl-4-[5-(1H-1,2,4-triazol-5-ylsulfanyl)furan-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
methyl 1-(2-methoxyethyl)-2-oxo-3-(pyrimidin-2-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
methyl 3-(5-ethyl-1,2-oxazole-3-carbonyl)-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
8-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}-1-oxa-8-azaspiro[4.6]undecan-9-one
4-(1-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-3-fluoro-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[(1R,2R,3R,5S)-2,6,6-trimethylbicyclo[3.1.1]heptan-3-yl]propanamide
1-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propan-1-one
N-[3-(1H-indol-2-yl)phenyl]-1-propanoylpiperidine-4-carboxamide
5-oxo-1-phenyl-N-(pyrimidin-4-ylmethyl)-2,5-dihydro-1H-pyrazole-3-carboxamide
5-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-(2-phenoxyethyl)azepan-2-one
(1S,5R)-6-(pyridazine-3-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]pyrrolidin-2-one
3-fluoro-N-[(7-{[5-(methoxymethyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzamide
3-hexyl-8-(1H-pyrrole-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3R,5S)-N-[(2-methoxyphenyl)methyl]-5-(morpholin-4-ylmethyl)piperidine-3-carboxamide
2-[9-(1-methyl-1H-pyrazole-4-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid