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1-[4-({[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
4-(piperidin-1-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}butanamide
N-{2-[2-(methylsulfanyl)pyridine-3-carbonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(4-methoxyphenyl)ethan-1-one
N-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-3-hydroxypiperidine-1-carboxamide
1-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-3-(pyrazin-2-yl)propan-1-one
2-(4-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}morpholin-3-yl)acetamide
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]pyridin-2-amine
methyl (2S)-1-{[4-(2-phenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}pyrrolidine-2-carboxylate
10-methoxy-N-(3-methyl-1,2,4-thiadiazol-5-yl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carboxamide
[(2S)-1-(4-{[(2-fluorophenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidin-2-yl]methanol
1-{2-[(2-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-cyclohexyl-N-methylpiperidine-4-carboxamide
N-{1-[7-(2-ethylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-methylbenzamide
(2E)-3-(2-chlorophenyl)-N-({3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]prop-2-enamide
methyl (2S)-2-(3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamido)-3-methylbutanoate
5-methyl-4-[2-methyl-2-(morpholin-4-yl)propyl]-1-(3-methylphenyl)piperazin-2-one
(2S)-2-amino-1-(4-{[4-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)propan-1-one
4-cyclobutyl-N-[(1-methanesulfonylpiperidin-3-yl)methyl]-6-methylpyrimidin-2-amine
methyl 2-[3-(3-{pyrazolo[1,5-a]pyrimidin-3-yl}phenyl)-1H-pyrazol-1-yl]acetate
3-{1-[3-(methylsulfanyl)propanoyl]piperidin-4-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
3-{5-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazol-5-yl]-3-methyl-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)propanamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}acetic acid
3-{4-[(dimethylamino)methyl]-4-hydroxyazepane-1-carbonyl}-1,2-dimethyl-1H-indol-5-ol
2-ethoxy-5-(2-{[(1S,2S)-2-hydroxycyclohexyl]amino}pyrimidin-4-yl)benzoic acid
N-methyl-1-(propan-2-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
methyl 2-(4-{[2-(dimethylamino)-6-methylpyrimidin-4-yl]amino}piperidin-1-yl)acetate
3-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[3-(1H-imidazol-1-yl)propyl]benzamide
2-methoxy-2-phenyl-N-[1-(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
2-(morpholin-4-yl)-1-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-6-ethyl-N,2-dimethylquinoline-4-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(N-methylmethanesulfonamido)ethyl]-1H-pyrazole-3-carboxamide
(2S)-2-[5-(4-methoxy-2-methylphenyl)-4-phenyl-1H-imidazol-1-yl]-4-(methylsulfanyl)butan-1-ol
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
N-[(1S,2R)-2-aminocyclobutyl]-4-(2,3-dihydro-1H-isoindol-2-yl)butanamide
4-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-1-(1H-indazol-6-yl)piperazin-2-one
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-[2-(furan-2-yl)-2-oxoacetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-{7-[(2,6-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
(2S,4R)-1-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-4-acetamido-N,N-diethylpyrrolidine-2-carboxamide
4-(6-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl)morpholine
N-(2-hydroxyethyl)-2,7-dimethyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyridine-3-carboxamide
4-({1-[5-(oxolan-2-yl)thiophene-2-carbonyl]piperidin-4-yl}oxy)pyridine
3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[3-(trifluoromethoxy)phenyl]methyl}propanamide
1-[(2R)-oxolane-2-carbonyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
4-{[1-(1-methyl-1H-indole-6-carbonyl)azetidin-3-yl]oxy}benzoic acid
N-[2-(benzylsulfanyl)ethyl]-1-methylazepane-2-carboxamide
N-benzyl-5-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{2-[({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]ethyl}piperidin-4-ol
N-ethyl-N-methyl-3-{[1-(pyrazin-2-yl)propan-2-yl]sulfamoyl}benzamide
1-(carbamoylmethyl)-N-{[1-(2-fluorophenyl)cyclopentyl]methyl}piperidine-3-carboxamide