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methyl (2S,4R)-4-(5-chloro-3-methyl-1H-indole-2-amido)-1-[(3-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxylate
N-[(3,4-difluorophenyl)methyl]-3-{1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-3-yl}propanamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-[2-(4-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]acetamide
N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-3-(2-oxopyrrolidin-1-yl)benzamide
{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}(2-methylpropyl)amine
2-(cyclohex-1-en-1-yl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]acetamide
(2-fluoro-5-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenyl)methanol
7-(1H-indole-2-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-methyl-9-{[3-(prop-2-en-1-yl)-4-(prop-2-en-1-yloxy)phenyl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
(1S,5R)-3-[4-(1H-pyrazol-4-yl)butanoyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
6-[(2-fluorophenyl)methoxy]-4-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
[(2S,4R,5R)-4-{[(5-ethylpyrimidin-2-yl)amino]methyl}-5-(2-fluorophenyl)-1-methylpyrrolidin-2-yl]methanol
ethyl 4-{1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carbonyl}piperazine-1-carboxylate
2-{4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-{2-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
4-(5-ethyl-2-methylpyrimidin-4-yl)-2-(trifluoromethyl)morpholine
3-ethyl-1-(2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-1,3-oxazole-4-carbonyl)piperidin-3-ol
N-[3-(methylsulfanyl)propyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
3-(4-chlorophenyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
methyl 4-(1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)piperazine-1-carboxylate
{4-benzyl-1-[3-(2-fluorophenyl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}methanol
3-chloro-N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-phenylethan-1-ol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-3-(thiophene-2-carbonyl)piperidine
1-(2-methanesulfonylethyl)-4-phenyl-5-(2,4,5-trifluorophenyl)-1H-imidazole
1-(dimethylamino)-2-[4-(3-methylbut-2-en-1-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-2-ol
1-(2,3-dimethylphenyl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-amine
N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
methyl 3-[(3-chlorophenyl)methyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3-methyl-1,2-oxazole-5-carbonyl)piperidine
3-[2-(4-hydroxypiperidin-1-yl)ethyl]-1-{4-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}urea
6-[(2,5-dimethoxyphenyl)methyl]-N-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
2-(4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}-6-methylpyrimidin-2-yl)phenol
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-1,4-diazepan-5-one
3-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-[3-(1,3-oxazol-5-yl)phenyl]urea
1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
3-{6-[(2-fluorophenyl)methoxy]-4-(2-methylpropyl)-3-oxo-1,4-diazepane-1-carbonyl}-1,2,5,6,7,8-hexahydroquinolin-2-one
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
2-{3-[2-amino-3-cyano-6-(2,2-dimethylcyclopropyl)-5-methylpyridin-4-yl]phenoxy}acetamide
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-2-ethyl-N,4-dimethyl-1,3-oxazole-5-carboxamide
2-butyl-8-(2,5-difluorobenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{[(4-fluoro-3-methylphenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(dimethyl-1,2-oxazol-4-yl)acetamide
1-[5-methoxy-2-({[3-(methylsulfanyl)propyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
N-butyl-N,5-dimethyl-4-{[3-(2-oxopyrrolidin-1-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
methyl 2-{[4-(hydroxymethyl)-4-(oxan-2-ylmethyl)piperidin-1-yl]sulfonyl}benzoate
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2,2-dimethyloxane-4-carboxamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
2-(4,6-dimethyl-1-benzofuran-3-yl)-1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]ethan-1-one