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2-(adamantan-1-yl)-1-[4-(pyrrolidin-1-yl)piperidin-1-yl]ethan-1-one
methyl 3-{[5-(5-chloro-2-fluorobenzoyl)-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
2,3-dimethyl-7-[4-(3-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)piperidine-1-carbonyl]-1H-indole
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-5-methyl-5-phenylpiperidin-2-one
4-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-4-oxobutanoic acid
(2S,4R)-N-[2-(dimethylamino)ethyl]-1-[(4-fluorophenyl)methyl]-4-[(4-methylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carboxamide
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]benzamide
N-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-2-(pyridin-3-ylmethyl)pyrrolidine-1-carboxamide
2-cyclopentyl-1-{9-[(1-methylpiperidin-4-yl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl}ethan-1-one
1-cyclohexyl-4-[6-(thiophen-3-yl)pyridine-3-carbonyl]-1,4-diazepane
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]-3-(3-ethoxypropyl)urea
2-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
1-[3-(1H-imidazol-1-yl)propyl]-5-(4-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazole
2,4-difluoro-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]benzamide
5-methyl-N-[2-(4-methylmorpholin-2-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
2-[(4-cyclopentyl-1,4-diazepan-1-yl)methyl]quinolin-4-ol
1-methyl-N-({8-[(4-methylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1H-pyrazole-3-carboxamide
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]acetamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-methylthieno[3,2-d]pyrimidin-4-amine
2-(2H-1,3-benzodioxol-5-yl)-8-methoxy-5-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-[4-(furan-2-yl)phenyl]-1-[3-(methylsulfanyl)propyl]piperidine-3-carboxamide
2-amino-6-(7-methoxy-1-benzofuran-2-yl)-4-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-N-methyl-N-(2-phenylethyl)piperidin-3-amine
6,7-dimethoxy-2-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-[2-(dimethylamino)-4-{[2-(pyridin-4-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
4-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-N-(1,2,3-thiadiazol-5-yl)benzamide
[(4-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl](oxan-4-ylmethyl)amine
4-(pyrrolidine-1-carbonyl)-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-{[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]methyl}benzoic acid
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-(oxolan-2-ylmethoxy)-4-[4-(1H-pyrazol-1-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 5-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
5-(piperidin-1-yl)-2-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,3-dihydropyridazin-3-one
(3aR,5R,6S,7aS)-2-{[3-(pyridin-2-yl)phenyl]methyl}-octahydro-1H-isoindole-5,6-diol
N-(2H-1,3-benzodioxol-5-yl)-6-[4-(1H-imidazol-1-yl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
7-(2,2-dimethylcyclopropanecarbonyl)-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl 3-{[4-(3-chlorothiophene-2-carbonyl)-7-oxo-1,4-diazepan-1-yl]methyl}benzoate
4-methoxy-4-phenyl-1-[3-(piperidin-3-yl)benzoyl]piperidine
1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
2-(2-hydroxyethyl)-9-[(4-methoxy-2-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}(4,4,4-trifluorobutan-2-yl)amine
N-{[7-(2,3-dimethoxybenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}furan-2-carboxamide
3-(2,4-dimethoxybenzoyl)-1-[(2E)-2-methylbut-2-en-1-yl]piperidine
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-5-phenylpentanamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-cyclopropyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-3-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]acetamide
2-(4-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperazin-1-yl)-1-(morpholin-4-yl)ethan-1-one
4-methyl-2-{2-[2-(thiophen-3-yl)-1H-imidazol-1-yl]ethyl}-6-(trifluoromethyl)pyrimidine
N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-3-(pyridin-3-yl)propanamide