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6-{[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-4-yl]amino}-2-methylheptan-2-ol
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[3-(1H-pyrazol-1-yl)propyl]propanamide
(3R)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(3,4-dimethylphenyl)-1-[3-(1H-imidazol-2-yl)benzoyl]piperidin-3-amine
2-methyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[2-(methylsulfanyl)ethyl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(pyridin-2-ylmethyl)piperazine
3-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-1-(2-methoxyethyl)-6-methyl-1,2-dihydroquinolin-2-one
1-{[(3R,4R)-1-(8-chloroquinolin-2-yl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
methyl 1-(2-methoxyethyl)-3-(2-phenylacetamido)-5-(propylamino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-chlorophenyl)urea
{1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-3-methylpiperidin-3-yl}methanol
N,N-diethyl-3-({[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)pyridin-2-amine
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-2-(pyrrolidine-1-carbonyl)piperazine
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-[(4-methylphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(dimethylamino)-1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]ethan-1-one
ethyl 1-(1-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)piperidine-3-carboxylate
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-5-methylpiperidin-2-one
1-[3-(morpholin-4-yl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-phenyl-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1,2,4-triazin-3-amine
methyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})(oxolan-3-ylmethyl)amine
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-methoxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
ethyl 2-[4-(4-fluorobenzenesulfonyl)-1-(3-methylbutyl)piperidin-4-yl]acetate
5-[1-(1H-indol-3-ylmethyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
3-[1-(1-cyclopropyl-5-oxopyrrolidine-3-carbonyl)piperidin-4-yl]benzonitrile
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
1-[cyclohexyl(methyl)amino]-3-[4-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1,2-oxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl 3-(4-{[3-(3-methylphenoxy)azetidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
4-{[(furan-2-ylmethyl)(pyridin-2-ylmethyl)amino]methyl}-6,7-dimethyl-2H-chromen-2-one
methyl 3-(2,4-difluorobenzoyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1R,5R)-6-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
6-(4-acetylphenyl)-N,N-dimethylpyridine-2-carboxamide
N-[(2R,3R)-1'-(5-methylthiophene-2-carbonyl)-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
(4-methylpentan-2-yl)({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amine
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
4-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}morpholine
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamide
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(pyrrolidine-1-carbonyl)piperidine
N-(2-{7-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
6-(1-methyl-1H-imidazol-2-yl)-N-[2-(pyridin-3-yloxy)propyl]pyridazin-3-amine
4-[4-(3-methoxyphenyl)piperazin-1-yl]pyrimidine-5-carboxylic acid
(3aR,7aS)-2-(5-ethyl-2-methylpyrimidin-4-yl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
3-hydroxy-N-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-3-(2-methylphenyl)pyrrolidine-1-carboxamide