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(2E)-1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)prop-2-en-1-one
(cyclohex-3-en-1-ylmethyl)({[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl})amine
1-[2-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-5-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)(pyridin-4-ylmethyl)amine
2-[4-(2,3-dimethoxy-5-methylphenyl)-1H-pyrazol-1-yl]ethan-1-ol
N-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methoxyethyl)-5-{[4-(trifluoromethyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[3-(4-ethylpiperazin-1-yl)propyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
4-(1-cyclopropyl-6-oxopiperidine-3-carbonyl)-1-(3-methoxyphenyl)piperazin-2-one
3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}propanamide
N-[1-(4-fluorophenyl)ethyl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-3-carboxamide
2-benzyl-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-1,3-thiazole-4-carboxamide
(3aS,6aS)-2-methyl-5-(1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(5-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)phenol
N-[(4-methylphenyl)(pyridin-4-yl)methyl]-3-(1,2-oxazinan-2-yl)propanamide
(1-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}piperidin-3-yl)methanol
3-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-1,5,6-trimethyl-1,2-dihydropyridin-2-one
N-{1-[1-(1H-indole-2-carbonyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,3-dimethylbutanamide
2-(1-ethyl-1H-imidazol-2-yl)-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
3-benzyl-8-[(3,4-difluorophenyl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{1-[(8-methylquinolin-5-yl)methyl]piperidin-2-yl}propan-1-ol
6-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(methylsulfanyl)pyrimidin-4-amine
2-{1-[(2-methylphenyl)methyl]-4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
1,4,6-trimethyl-3-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
3-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
methyl 3-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl](methyl)carbamoyl}benzoate
2-amino-8-(5-ethyl-2-methylpyrimidin-4-yl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)acetic acid
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[(5-methylfuran-2-yl)methyl]pyridin-2-amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-{2-[2-(2-methoxyethyl)piperidin-1-yl]-2-oxoethyl}-3-phenylpyrrolidine-2,5-dione
5-cyclopropyl-N-(3-ethoxypropyl)-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-ethyl-5-{2-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-oxoethyl}-6-methyl-3,4-dihydropyrimidin-4-one
2,3-dimethoxy-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]benzamide
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-3-methyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
3-{2-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-2-oxoethyl}-1,3-thiazolidine-2,4-dione
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[1-(4-methylphenyl)piperidin-4-yl]pyrrolidin-3-yl]methanol
5-[4-(4-methoxyphenyl)-3-oxopiperazine-1-carbonyl]pyridine-2-carbonitrile
3-{5-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-(3,3-diphenylpropyl)-6-(pyridin-3-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
4-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]morpholine-2-carboxylic acid
ethyl 4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carboxylate
N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]-1H-pyrazole-4-carboxamide
1-[1-(cyclohexylmethyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
(5S,9aS,9bS)-5-[4-methoxy-3-(methoxymethyl)phenyl]-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-[1-(2-hydroxyethyl)-1H-pyrazol-4-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-3-methylbut-2-enamide
3-[(7-fluoro-4-methylquinolin-2-yl)amino]propan-1-ol
2-(furan-2-yl)-1-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]pyrrolidine
2-fluoro-N-{[8-(thiophene-3-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide