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methyl 4-{5-[({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl)amino)methyl]-1,2,4-oxadiazol-3-yl}benzoate
2-ethyl-N-[3-(1H-imidazol-1-yl)propyl]-1-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-[4-(2-methyl-1,3-thiazole-4-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
benzyl[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]methylamine
(2S,4R)-1-[(2-hydroxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-(quinoxalin-6-yl)pyrrolidine-2-carboxamide
3-[3-(4-fluorophenyl)phenyl]propanamide
(3R)-1-{[5,8-dimethoxy-2-(2-methoxyphenyl)quinolin-3-yl]methyl}pyrrolidin-3-ol
(1R,5R)-6-[(3,5-dichloropyridin-4-yl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(1,3-dimethyl-1H-pyrazol-5-yl)-5-{[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}-1,3-thiazol-2-amine
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-acetamido-3-methylbutanamide
N-({1-[(E)-2-phenylethenesulfonyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
4-{[2-hydroxy-5-(pyridin-2-yl)phenyl]methyl}piperazine-1-carbaldehyde
3-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-N-[(2-fluorophenyl)methyl]propanamide
N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-4-hydroxy-2-(thiophen-2-yl)pyrimidine-5-carboxamide
1-cyclopentyl-3-(2-fluorophenyl)-3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
N-{[7-fluoro-5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}naphthalene-2-carboxamide
N-ethyl-N-[2-(2-fluorophenoxy)ethyl]-2-methylfuran-3-carboxamide
1-(2-phenoxyethyl)-4-(piperidin-3-ylmethyl)piperazine
ethyl 1-benzyl-5-(4-methyl-1,3-oxazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]-4-(4-methyl-1H-pyrazol-3-yl)piperidine
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}acetamide
6-[3-(5-methyl-2-{[2-(morpholin-4-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidine-1-carbonyl]-1H-indole
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-(2-{[2-(morpholin-4-yl)ethyl]carbamoyl}phenyl)-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-({7-[2-(2-methoxyphenoxy)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenoxypropanamide
N-({7-[2-(3-fluorophenyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
(oxolan-2-ylmethyl)({[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl})(pyridin-2-ylmethyl)amine
N-[2-(3-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy)propyl]pyridine-2-carboxamide
2-(dimethylamino)-7-(4,4,4-trifluorobutanoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
N-methyl-N-(1,3-thiazol-2-ylmethyl)-3-[({[4-(trifluoromethyl)phenyl]methyl}amino)methyl]-6H,7H,8H-cyclopenta[g]quinolin-2-amine
2-[5-(6-methylpyridin-2-yl)-4-phenyl-1H-imidazol-1-yl]propane-1,3-diol
N,2,2-trimethyl-4-oxo-N-[1-(3-phenylpropyl)piperidin-3-yl]-3,4-dihydro-2H-pyran-6-carboxamide
8-[(3,4-difluorophenyl)methyl]-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{2-[3-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-1-ethyl-3-(2-methylphenyl)pyrrolidine-2,5-dione
N-(dicyclopropylmethyl)-N-methyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
5-[1-(3,5-dimethoxybenzoyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2-[1-(4-chlorophenyl)cyclobutanecarbonyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)furan-2-carboxamide
2-(4-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)-1,3-benzothiazole
2-cyclopentyl-N-[1-methyl-2-(oxolan-2-yl)-7-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H-1,3-benzodiazol-5-yl]acetamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[3-(quinolin-8-yl)-1H-indazol-1-yl]acetamide
7-(2,2-dimethylpropyl)-2-[3-(1H-pyrazol-1-yl)propyl]-2,7-diazaspiro[4.5]decan-6-one
N-(2-{1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]piperidin-2-yl}ethyl)acetamide
3-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-6-(trifluoromethyl)pyridin-2-ol
3-(4-phenylbenzoyl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine
N-[2-methyl-1-(7-{[4-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]pyridine-2-carboxamide