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1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(3,4-difluorophenyl)ethan-1-one
N-cyclopropyl-N-[(2E)-3-phenylprop-2-en-1-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
(2S,4S)-4-amino-1-(3-cyclobutaneamido-4-methylbenzoyl)-N-methylpyrrolidine-2-carboxamide
5-fluoro-2-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}-3-methyl-1H-indole
5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1-methyl-1H-1,2,3-benzotriazole
5-(propan-2-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1,2-oxazole-3-carboxamide
3-(4-fluoro-3-methylphenyl)-6-(5-methylpyrazine-2-carbonyl)-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
4-ethyl-N-{2-[1-(propan-2-yl)piperidin-3-yl]ethyl}-1,2,3-thiadiazole-5-carboxamide
1-{2-[4-(ethanesulfonyl)piperazin-1-yl]pyrimidin-4-yl}pyrrolidin-3-ol
N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]thiolan-3-amine
2-benzyl-N-methyl-N-(1,2-oxazol-5-ylmethyl)-1,3-thiazole-4-carboxamide
4-(3,4-difluorophenyl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
7-(1-benzothiophen-3-yl)-4-[(1-methyl-1H-imidazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 5-{[(3-fluorophenyl)methyl]amino}-3-(furan-2-amido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
({4-cyclopropyl-5-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
4-(oxolane-3-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(4aR,7aS)-1-butyl-4-[(2-phenyl-1,3-oxazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methyl-5-[3-methyl-1-(3-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]phenol
2-(4-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperazin-1-yl)pyridine-4-carboxamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[3-(1H-imidazol-1-yl)propyl](pyridin-3-ylmethyl)amine
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{2-[({4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}methyl)amino]ethyl}methanesulfonamide
2-(4-{[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]amino}-6-methylpyrimidin-2-yl)phenol
1-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3-[3-methyl-1-(2-methylpropyl)-1H-pyrazol-5-yl]urea
2-{4-phenyl-1-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-1H-imidazol-5-yl}quinoline
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyridine-3-carboxylic acid
4-[4-(2-ethylpiperidine-1-carbonyl)piperidin-1-yl]-2-(pyridin-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
ethyl 4-benzyl-1-[(5-ethylfuran-2-yl)methyl]piperidine-4-carboxylate
4,5-dimethyl 1-[(3S,5S)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
3-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}-N-[(3-methoxyphenyl)methyl]piperidine-1-carboxamide
ethyl 3-(3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamido)propanoate
1-(4-tert-butylbenzoyl)-4-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,4-diazepan-5-one
N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopropanecarboxamide
2-[(furan-2-ylmethyl)({[4-(pyrimidin-2-yloxy)phenyl]methyl})amino]butan-1-ol
N-(4-chloro-3-methylphenyl)-2-({2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}amino)acetamide
N-[(3R,4R)-3-hydroxy-1-[(3E)-4-methylhex-3-en-1-yl]piperidin-4-yl]pyridine-2-carboxamide
5-ethyl-2-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}pyridine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-[4-(1-benzothiophen-3-yl)-2-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy]acetamide
1-[4-(cyclopropylmethyl)piperazin-1-yl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
1-{[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}-3-propoxypiperidine
3,5-dichloro-N,4-dimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
(3aR,7aS)-2-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-{1-[(5-chloro-1-benzothiophen-3-yl)methyl]-1H-imidazol-2-yl}-1-methyl-1H-imidazole
(1R,7S)-6-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-3-(2-ethylbutyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-[3-ethoxy-4-(prop-2-en-1-yloxy)benzoyl]imidazolidin-4-one
N-{[8-(2H-1,3-benzodioxol-5-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}pyridine-3-carboxamide
2-[3-oxo-9-(3,3,3-trifluoro-2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
5-[({[3-(2-{4-[4-(1H-imidazol-1-yl)benzoyl]piperazin-1-yl}ethoxy)phenyl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
3-(diphenylmethyl)-N-(oxan-4-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide