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N-{1-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanoyl]piperidin-4-yl}methanesulfonamide
5-(2-fluorophenyl)-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-[2-({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
1-[(2-methoxyphenyl)methyl]-6-oxo-N-[2-(2-oxoimidazolidin-1-yl)ethyl]piperidine-3-carboxamide
3-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-1H-indazole
1-{2-oxo-2-[1-(pyridin-3-yl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl]ethyl}piperidine-4-carboxamide
3-(3,4-difluorophenyl)-5-(3-fluoro-4-methoxybenzoyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-{[3-(cycloheptyloxy)-4-methoxyphenyl]methyl}-N-cyclopropylcyclobutanecarboxamide
8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-[4-(trifluoromethyl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(1,3-dihydroxy-2-methylpropan-2-yl)-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-(1-{5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-phenyl-1H-imidazol-1-yl}ethyl)-1H-1,2,4-triazole
1-[(3-chlorophenyl)methyl]-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(2-amino-4-methyl-1,3-thiazol-5-yl)-1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]ethan-1-one
3-[1-(8-fluoroquinoline-2-carbonyl)piperidin-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
3-({3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)-1,2-dihydroquinolin-2-one
5-methyl-5-[1-(quinolin-6-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
N-(1,4-dioxan-2-ylmethyl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
1-[1-(4-chlorobenzoyl)piperidin-3-yl]-3-phenylpropan-1-one
N-{2-[1-(4-chlorophenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-N-methylmethanesulfonamide
N-(1-{7-[(3,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
1-ethyl-N-[3-(3-fluorophenyl)phenyl]piperidine-4-carboxamide
4-[3-(ethoxycarbonyl)-3-[(2-fluorophenyl)methyl]piperidine-1-carbonyl]pyridin-1-ium-1-olate
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}oxolane-2-carboxamide
2-methoxy-1-(3-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carbonyl}piperidin-1-yl)ethan-1-one
3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(pyridin-4-yl)propan-2-yl]propanamide
6-methyl-4-[4-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
(1S,6R)-9-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}-3,9-diazabicyclo[4.2.1]nonane
methyl (2S,4S)-1-benzyl-4-(2-methoxybenzamido)pyrrolidine-2-carboxylate
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-(2-methoxyphenyl)propan-1-one
2-[4-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-1-yl]-N-(propan-2-yl)acetamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-N,N-diethyl-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
6-[4-(benzyloxy)-3-fluorophenyl]-N,N-dimethylpyridine-2-carboxamide
methyl (2S)-1-{2-[4-(4-{[2-(pyridin-3-yloxy)ethyl]amino}piperidin-1-yl)phenyl]acetyl}pyrrolidine-2-carboxylate
N,N-diethyl-2-({4-[2-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetyl]-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl}oxy)acetamide
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
2-(1-methyl-1H-pyrrol-3-yl)-1-[1-(pyridin-2-ylmethyl)-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}isoquinoline-5-carboxamide
3-{[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]sulfamoyl}-N-(pentan-2-yl)benzamide
6-(cyclopropylmethoxy)-4-[2-(2,5-dimethoxyphenyl)acetyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
3-methyl-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
(4aR,8aS)-1-[2-(diethylamino)ethyl]-6-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]-decahydro-1,6-naphthyridin-2-one
methyl 1-[2-hydroxy-3-(4-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenoxy)propyl]piperidine-4-carboxylate
4-[4-(2-phenylpyrimidin-4-yl)piperidine-1-carbonyl]-1,2-dihydrophthalazin-1-one
N-[(2R,3R)-2-hydroxy-1'-[(2-hydroxy-3-methoxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
3-[1-(1-methylazepane-2-carbonyl)piperidin-4-yl]-N-phenylpropanamide
2-[3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)phenoxy]acetic acid
N-(1,4-dioxan-2-ylmethyl)-4-(4-methylpiperazin-1-yl)benzamide