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{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}[1-(2-methoxyphenyl)ethyl]methylamine
1-[6-(pyridin-3-yl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
N-[2-(benzyloxy)ethyl]-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
[(3R,5R)-1-(2,6-difluoro-3-methoxybenzoyl)-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
N-cyclopentyl-5-{1-[2-(pyridin-3-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]acetamide
methyl 3-[(cyclopropylformamido)methyl]-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
1-methyl-3-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
3-[(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-3-yl)methyl]benzoic acid
ethyl 4-[1-(2-methoxyphenyl)-1H-pyrazole-4-amido]piperidine-1-carboxylate
4-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-2-(methylsulfanyl)-1,3-thiazole
4-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}sulfonyl)benzoic acid
1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
3-(diphenylmethyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,2-oxazole-5-carboxamide
(2S,4S)-4-amino-N-ethyl-1-[2-(methylamino)benzoyl]pyrrolidine-2-carboxamide
N-(1-{7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1-methylpiperidine-4-carboxamide
2-[9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
7-[6-(4-hydroxypiperidin-1-yl)pyrimidin-4-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-{4-[(4-ethoxyphenyl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
2-{[(1S,4S)-5-benzyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]methyl}-8-chloroquinolin-4-ol
3-(oxolan-3-yl)-5-(4-propoxyphenyl)-1,2,4-oxadiazole
1-(2,4-dimethoxybenzoyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
2-methoxy-5-(1-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-imidazol-2-yl)pyrimidine
ethyl 4-[6-(2,5-dimethoxyphenyl)-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridine-3-amido]piperidine-1-carboxylate
3-[(cyclopentylamino)methyl]-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
methyl[(5-methyl-3-phenyl-1,2-oxazol-4-yl)methyl][2-(1H-pyrazol-4-yl)ethyl]amine
5-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1,2-dihydropyridin-2-one
5-(naphthalen-1-ylmethyl)-5-{3-oxo-3-[2-(pyridin-3-yl)piperidin-1-yl]propyl}pyrrolidin-2-one
3-(4-methoxypiperidine-1-carbonyl)-N-(1H-pyrazol-3-ylmethyl)benzene-1-sulfonamide
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
dimethyl(2-{2-[3-(1H-pyrazol-3-yl)phenyl]phenoxy}ethyl)amine
2-cyclopropyl-1-{5-[5-(4-fluorophenyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}ethan-1-one
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyrrolidin-1-yl)ethan-1-one
2-[2-fluoro-3-(pyrrolidin-1-ylmethyl)phenoxy]-5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
1-(2,3-dihydro-1-benzofuran-2-ylmethyl)-1-methyl-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
(1S,5R)-3-[(5-butylthiophen-2-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,9S)-5-amino-3-(4-fluoro-3-methylphenyl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-benzyl-N5-ethyl-N3-methyl-4-oxo-N3-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
4-(3-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyrimidin-2-amine
5-methyl-5-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
N-ethyl-5-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}pyrimidin-2-amine
N-(1-{7-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
6-methyl-2-[(2-methylphenyl)methyl]-N-(1,2-oxazol-3-ylmethyl)-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
N-methyl-N-(propan-2-yl)-2-[2-(1H-pyrazol-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
methyl 5-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
3-(4-chlorophenyl)-1-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine
ethyl 4-{[(1,3-benzothiazol-5-yl)carbamoyl]amino}piperidine-1-carboxylate
N5-[(8-methoxyquinolin-5-yl)methyl]-N5,N6,N6-trimethyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-[(2R,3R)-2-methoxy-1'-{2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide