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1-(2-methylpropyl)-4-[3-(1H-pyrazol-1-yl)benzoyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
3-(1-{[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[7-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopent-1-ene-1-carboxamide
methyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-1-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]propan-1-one
4-cyclopentyl-11-[(3-ethoxypropyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-ethyl-4-(2-{3-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)piperazine-2,3-dione
1-(4,7-dimethylquinazolin-2-yl)-N-[(3-methoxyphenyl)methyl]-N-methylpiperidine-3-carboxamide
(2R,3R,6R)-3-(4-fluorophenyl)-5-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-3-carbonyl]morpholine
(3S,9aR)-3-benzyl-8-[(5-chlorothiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-(7-{[4-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclobutanecarboxamide
(3S,9aR)-3-[(2S)-butan-2-yl]-8-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N4-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N2,N2-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
3-acetamido-N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)thiophene-2-carboxamide
(4aS,8aS)-2-[5-(morpholin-4-ylmethyl)pyridin-2-yl]-decahydro-2,7-naphthyridin-4a-ol
1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
5-methyl-2-[(pyridin-2-ylmethyl)sulfanyl]-4-[1-(thiophene-2-carbonyl)piperidin-3-yl]pyrimidine
7-[(2,4-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
({4-[(2-chloro-3,4-dimethoxyphenyl)methyl]-1,4-oxazepan-6-yl}methyl)dimethylamine
6-(2-fluorophenyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(pyridin-3-ylmethyl)amine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)cyclopentanecarboxamide
(4S)-N-[(3-fluorophenyl)methyl]-4-hydroxy-3,3,4-trimethylpiperidine-1-carboxamide
N3-butyl-N5-[(3,5-difluorophenyl)methyl]-1-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-methoxy-2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
[(3R,4R)-1-{[3-(furan-2-yl)phenyl]methyl}-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}ethane-1-sulfonamide
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-1-(methoxymethyl)cyclobutane-1-carboxamide
N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}-2-(2-methyl-1H-imidazol-1-yl)propanamide
5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-N-methyl-N-[(5-methylfuran-2-yl)methyl]pyridin-2-amine
7-(3-chlorophenyl)-4-[2-(oxolan-3-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-pyrazole-5-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-ylmethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(dimethyl-1,2-oxazol-4-yl)-3-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)benzamide
3-(1H-1,3-benzodiazol-1-yl)-N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
N-ethyl-N-(1-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-2-phenylethyl)oxane-4-carboxamide
N'-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N'-(2-methoxyethyl)butanediamide
1-cyclohexyl-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(2,4-difluorophenyl)-1-[1-(5-fluoro-1H-indole-2-carbonyl)piperidin-4-yl]ethyl]-N-methylpropanamide
3-[(2,3-dimethoxyphenyl)methyl]-5-[1-(4-methoxybenzoyl)piperidin-4-yl]-5-methylimidazolidine-2,4-dione
1-{4-[3-oxo-3-(4-phenylpiperazin-1-yl)propyl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(3aS,6aS)-2-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
(1R,5R)-6-[2-(2,4-difluorophenoxy)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
({3-[(1-cyclohexanecarbonylpiperidin-4-yl)oxy]phenyl}methyl)(methyl)(thiophen-3-ylmethyl)amine
6-{[2-(1-hydroxycyclopentyl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
2-[2-(3-chloro-4-hydroxyphenyl)acetamido]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-methyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
1-(4,7-dimethylquinazolin-2-yl)-N-[2-(2-fluorophenyl)ethyl]piperidine-4-carboxamide