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5-[1-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-3-yl]-4-methyl-N-[(3-methylthiophen-2-yl)methyl]-1,3-thiazol-2-amine
2-(phenylsulfanyl)-N-[1-({[2-(pyridin-4-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]acetamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-[2-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
2-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-(3-hydroxy-2,2-dimethylpropyl)-3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}propanamide
1-(cyclohexylmethyl)-3-[4-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
4-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-1-phenylpiperazin-2-one
3-[(3R,4S)-4-(dimethylamino)-1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)piperidin-3-yl]propan-1-ol
N,4-dimethyl-5-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,3-thiazol-2-amine
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-6-(methoxymethyl)pyridine-2-carboxamide
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]furan-3-carboxamide
(3S)-1-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}pyrrolidin-3-ol
N-methyl-2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
3-[5-({3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}methyl)-1,3,4-oxadiazol-2-yl]pyridine
4-[(3-hydroxyphenyl)methyl]-N-[2-(propylsulfanyl)phenyl]piperazine-1-carboxamide
N-{2-[4-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]ethyl}aniline
N-(2,3-dihydro-1H-inden-2-yl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-4-carboxamide
2-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)quinoline
N-({7-[(2E)-3-(3,5-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-sulfonamide
2-[3-(4-methoxyphenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]acetamide
4-chlorophenyl (7S,9aR)-7-[(benzyloxy)methyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N-methyl-2-[(1-methyl-1H-indol-3-yl)sulfanyl]-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]acetamide
8-[(2-ethylpyrimidin-5-yl)methyl]-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
9-(cyclopropylmethyl)-1-methyl-4-(pyrimidin-2-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(4-ethoxyphenyl)methyl]piperidine
methyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
3-(3-amino-1H-indazol-1-yl)-5-(morpholine-4-sulfonyl)benzoic acid
[(3R,4R)-1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
ethyl 3-{[3-(2-phenylpropyl)-1,2-oxazol-5-yl]formamido}propanoate
2-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-dimethylbenzamide
1-[3-(4-fluorophenyl)pyrrolidin-1-yl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propan-1-one
4-({[2-amino-6-(propan-2-yl)pyrimidin-4-yl]amino}methyl)phenol
(2S,4S)-4-amino-1-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-N-methylpyrrolidine-2-carboxamide
1-[(1-methyl-1H-imidazol-5-yl)methyl]-4-(2-phenylethyl)piperidine
2-[(3S,4R)-3-cyclopropyl-4-(oxane-4-amido)pyrrolidin-1-yl]acetic acid
2-chloro-N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-N-(2-hydroxyethyl)pyridine-4-carboxamide
1-[2-(ethylsulfanyl)phenyl]-3-{[1-(methoxymethyl)cyclopentyl]methyl}urea
1-(2-methylpropyl)-8-(naphthalen-2-ylmethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-({1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}methyl)-3-(propan-2-yl)urea
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]propanamide
N-(1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-cyclopentyl-3-(1H-imidazol-1-yl)-N-(3-phenylprop-2-yn-1-yl)propanamide
4-{[(1R,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2,1,3-benzoxadiazole
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(1H-pyrazol-1-yl)benzamide
1-{3-[4-({[(5-fluoro-2-methylphenyl)methyl]amino}methyl)-2-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
N-(1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
(4aS,8aR)-4a-(hydroxymethyl)-N-[3-(trifluoromethyl)phenyl]-decahydro-1,6-naphthyridine-6-carboxamide
1-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)pyrrolidine
3-chloro-5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]pyridine