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1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
N3-methyl-4-oxo-1-(3-phenylpropyl)-N5-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
benzyl({[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})ethylamine
4-chloro-1-methyl-3-[3-methyl-1-(3-methylbutyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrazole
1-cyclopentyl-3-(3-fluorophenyl)-3-{2-[4-(2-fluorophenyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
5,8-dimethyl-2-({[2-(1,3-thiazol-4-yl)ethyl]amino}methyl)quinolin-4-ol
1-(cyclohexylmethyl)-6-oxo-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
2-ethyl-N-[2-(2-phenoxyethoxy)phenyl]pyrimidine-5-carboxamide
1-(1-{5-[(dimethylsulfamoyl)amino]-1-methyl-2-(2-methylpropyl)-1H-1,3-benzodiazole-7-carbonyl}piperidin-3-yl)ethan-1-one
(2R,6S)-4-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]-2,6-dimethylmorpholine
2-[(4aS,8aR)-2-oxo-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-6-yl]pyridine-4-carbonitrile
2-butyl-5-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidine-1-carbonyl}-1,3-benzoxazole
N-cyclopentyl-4-(4-{[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]amino}piperidin-1-yl)benzamide
1-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}-3-methylpentan-1-one
1-[(3-methoxyphenyl)methyl]-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-3-(1-methylpiperidin-2-yl)propanamide
N-{[7-(5-chloro-3-methyl-1H-indole-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-fluorobenzamide
methyl 5-({[3-(2-hydroxyethoxy)phenyl]methyl}amino)-3-(2-methoxyacetamido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{[2-(2-chloro-6-fluorophenyl)-1H-imidazol-1-yl]methyl}pyridine
9-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-6-oxa-9-azaspiro[4.5]decane
2-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-5-methylpyrazine
methyl[(2-methyl-1,3-oxazol-4-yl)methyl]{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(2S,4R,6S)-2-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-6-(2-methylpropyl)oxan-4-yl]acetamide
(1S,5R)-3-methyl-6-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[2-(propylsulfanyl)ethyl]benzamide
N'1-[(3R,4S)-1-(2-methanesulfonylethyl)-4-(propan-2-yl)pyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
ethyl 1-[5-acetamido-1-ethyl-2-(3-methoxyphenyl)-1H-1,3-benzodiazole-7-carbonyl]piperidine-4-carboxylate
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-2,4-dimethylpyrimidine
(2R)-2-{[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}hexanoic acid
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
9-(2-amino-5-methylpyrimidin-4-yl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
6,7-diethoxy-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-3-methyl-1-benzofuran-2-carboxamide
1-methyl-4-oxo-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-1,4-dihydroquinoline-3-carboxamide
ethyl 1-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-3-(2-methoxyethyl)piperidine-3-carboxylate
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}propane-2-sulfonamide
2-(1-ethyl-1H-pyrazol-4-yl)-N-[1-(pyridin-3-yl)propan-2-yl]quinoline-4-carboxamide
5-(pyridin-3-yl)-5-{1-[2-(1,3-thiazol-4-yl)acetyl]piperidin-4-yl}-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-(2,5-difluorobenzoyl)-1-(5-methylthiophene-2-carbonyl)piperidine
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
3-[4-(2,5-difluorophenyl)-1H-pyrazol-5-yl]-1-(2,2-dimethylpropyl)piperidine
2-chloro-9-methyl-3-{3-oxa-9-azaspiro[5.5]undecan-9-ylmethyl}-4H-pyrido[1,2-a]pyrimidin-4-one
N-[3-(4-methylbenzenesulfonamido)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-{4-[2-(phenoxymethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
(3S)-1-[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]pyrrolidin-3-ol
2-(1H-imidazol-2-yl)-N-methyl-N-(thiophen-3-ylmethyl)benzamide
3-{5-[(2R)-oxolan-2-yl]-1,2,4-oxadiazol-3-yl}-2-phenoxypyridine
3-methoxy-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,2-dihydropyridin-2-one
(3S,4R)-1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-(2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid