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4-(2,1,3-benzoxadiazol-4-ylmethyl)piperazine-1-sulfonamide
2-(4-chloro-1H-pyrazol-1-yl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]acetamide
3-(2H-1,3-benzodioxol-5-yl)-1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propan-1-one
1-{4-[2-(dimethylamino)ethyl]piperazin-1-yl}-2-(2,5-dimethylphenoxy)propan-1-one
1-[1-(4-fluorophenyl)cyclopropanecarbonyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-[1-(4-chlorobenzoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-(2-methylphenyl)-3-(1-{1-[2-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
4-(4-methyl-1,3-oxazole-5-carbonyl)-1-(2-methylpropyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-[(2,6-difluoro-3-methylphenyl)methyl]-5-[(dimethylsulfamoyl)amino]-1-methyl-2-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
4-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]benzene-1-sulfonamide
(3R,4R)-3-cyclopropyl-1-(5-fluoro-2-methylbenzoyl)-4-methylpyrrolidin-3-ol
1-(1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-3-methylbutan-1-one
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-methyl-N-(2-methylpropyl)acetamide
3-(3-methyl-1H-pyrazol-1-yl)-1-[4-(3-methylphenoxy)piperidin-1-yl]propan-1-one
8-[2-(dimethylamino)acetyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
5-(4-cyclobutyl-6-methylpyrimidin-2-yl)-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]ethan-1-one
1-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
2-{5-[(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)methyl]-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-1-yl}acetic acid
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1-propyl-1H-pyrazole-5-carboxamide
3-[3-({[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]amino}methyl)-1H-indol-1-yl]propanamide
methyl[(3-methyl-1H-indol-2-yl)methyl]{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(2,6-difluorophenyl)methyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
3-{1-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl](ethyl)(pyridin-4-ylmethyl)amine
6-{[3-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}pyridine-2-carboxylic acid
1-[(4-methoxyphenyl)methyl]-4-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperazin-2-one
8-[(3,4-dimethylphenyl)methyl]-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-methyl-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-1H-pyrazole-5-carboxamide
2-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-[3-(4-phenylpiperazine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-pyrazol-1-yl)propan-1-one
3-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-9-(1,2-oxazole-5-carbonyl)-3,9-diazaspiro[5.5]undecane
N-methyl-2-{4-[methyl(2-phenylethyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}-N-(propan-2-yl)acetamide
1-[3-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)phenyl]pyrrolidin-2-one
5-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)imidazolidine-2,4-dione
2-[1-(3-methylbutyl)-4-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-{1-[2-(3,5-difluorophenyl)acetyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
ethyl 4-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylate
(4aS,8aR)-6-[(4-methyl-1H-imidazol-5-yl)methyl]-1-[2-(5-methylfuran-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
[(2,4-dimethoxyphenyl)methyl]({[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl})amine
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(1H-pyrazol-1-yl)benzamide
3-(1H-1,3-benzodiazol-2-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}propanamide
2-acetamido-N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}acetamide
4-{2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}benzene-1-sulfonamide
4-{8-[3-(1H-imidazol-1-yl)butanoyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}butanoic acid
3-(but-2-yn-1-yl)-5-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
{3-[2-(1-cyclopentanecarbonylpiperidin-3-yl)-1H-imidazol-1-yl]propyl}dimethylamine
2-(cyclopropylmethyl)-8-[2-(3-oxopiperazin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one