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[(3R,4R)-4-(pyrrolidin-1-ylmethyl)-1-(quinoxaline-6-carbonyl)pyrrolidin-3-yl]methanol
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
2-amino-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-4-(3-hydroxyphenyl)pyridine-3-carbonitrile
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N-methyl-4-oxo-N-(pyridin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-[(1-methanesulfonylpyrrolidin-3-yl)methyl]benzamide
8-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
[(3R,4R)-4-[(dimethylamino)methyl]-1-[3-(4-fluorophenyl)benzoyl]pyrrolidin-3-yl]methanol
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[3-(trifluoromethoxy)phenyl]methyl}propanamide
methyl({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})[2-(pyridin-4-yl)ethyl]amine
2-(2H-1,3-benzodioxol-5-yl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-methyl-3-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-1-[3-(1,3-oxazol-5-yl)phenyl]urea
8-(1-benzylpiperidine-2-carbonyl)-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(ethoxymethyl)-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidine
1-[3-(morpholin-4-yl)propyl]-5-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)piperidin-2-one
7-(pyridine-3-carbonyl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-hydroxy-3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-{4-[1-(1,4-dithiepan-6-yl)pyrrolidin-3-yl]piperidin-1-yl}pyrimidine
1-(2,1,3-benzoxadiazol-5-ylmethyl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
1-benzyl-2-methyl-3-[2-(morpholin-4-yl)-2-oxoethyl]-4,5,6,7-tetrahydro-1H-indol-4-one
1-[4-(4-chlorophenoxy)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
(4aS,7aR)-1-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{[2-(benzyloxy)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
5-[3-(4-tert-butylphenyl)propyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
N-{[7-(furan-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(piperidin-1-yl)acetamide
5-(6-aminopyridine-3-carbonyl)-N-cyclopropyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-{1-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-[(1S)-2-(1H-imidazol-4-yl)-1-[1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]ethyl]acetamide
3-(2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine-4-carbonyl)-4,6-dimethyl-1,2-dihydropyridin-2-one
[(3R,4R)-1-(3-fluoro-4-methoxybenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-5-methyl-1-benzofuran-2-carboxamide
4-{4-[3-(3-methoxybenzoyl)piperidine-1-carbonyl]phenyl}-2-methylbut-3-yn-2-ol
5-[4-(4-methoxyphenyl)butan-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
1-(2-methylpropyl)-4-(3-phenoxypropanoyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
5-(4-acetylphenoxymethyl)-N-[phenyl(pyridin-4-yl)methyl]-1,2-oxazole-3-carboxamide
4-[4-ethoxy-3-methoxy-5-(prop-2-en-1-yl)phenyl]-3-methyl-4H,5H,6H,7H-[1,2]oxazolo[5,4-b]pyridin-6-one
1-(4-methyl-2-{9-oxa-2-azaspiro[5.5]undecan-2-yl}pyrimidin-5-yl)ethan-1-one
(2S,4R)-1-[(2,4-difluorophenyl)methyl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
(2E)-N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-(3-fluorophenyl)prop-2-enamide
1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-5-[5-(propan-2-yl)-1,3-oxazol-4-yl]-1H-1,2,4-triazole
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-methoxy-4-(2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-5-(5-methylfuran-2-yl)-N-(pyrazin-2-ylmethyl)-1,2,4-triazin-3-amine
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-(1,2,3,4-tetrahydronaphthalen-2-yl)urea
3-(cyclopropylmethyl)-5-[(4-fluorophenyl)methyl]-5-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}butanamide
2-(2-methyl-1,3-thiazol-4-yl)-1-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)ethan-1-one
2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(3,4-dimethoxyphenyl)methyl]acetamide
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}piperidine-3-carboxamide
N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
2-[2-methoxy-4-({2-methyl-2,7-diazaspiro[4.5]decan-7-yl}methyl)phenoxy]acetamide