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1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperazine
[(3S,5R)-1-(4-chloro-3-methylbenzoyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
5-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1-benzofuran-2-carboxamide
N-(adamantan-1-ylmethyl)-N-methyl-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(morpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-(1,3-benzoxazol-2-yl)-N-(1,3-dimethyl-1H-pyrazol-5-yl)piperazine-1-carboxamide
1-methyl-2-oxo-8-(4-oxo-4-phenylbutanoyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[4-(3-methylpiperidine-1-carbonyl)piperidin-1-yl]-2-(pyridin-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
8-methoxy-N-[1-(3-phenylpropyl)piperidin-3-yl]quinolin-2-amine
({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[2-(2-methyl-1H-indol-1-yl)ethyl]amine
(1S,2R)-1-{[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}-2,3-dihydro-1H-inden-2-ol
N-[3-(2-methoxyphenyl)propyl]-1,4-dithiepan-6-amine
(3R,4S)-N,N-dimethyl-1-[6-(piperidine-1-carbonyl)pyrazin-2-yl]-4-propylpyrrolidin-3-amine
1-(3-{[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}phenyl)ethan-1-one
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[2-(3-methylthiophen-2-yl)ethyl]acetamide
4-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-6-(2-methylpropyl)pyrimidin-2-amine
(4aS,8aR)-6-[(3-ethoxyphenyl)methyl]-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
4-methanesulfonyl-N-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]piperazine-1-carboxamide
1-[2-methoxy-5-({[(2-methoxyphenyl)methyl](methyl)amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
1-[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-N-methylpiperidine-3-carboxamide
4-({1-[(4-ethylphenyl)methyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl}methyl)morpholine
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}cyclobutanecarboxamide
2-(2,3-difluorophenoxymethyl)-N-(1H-indol-2-ylmethyl)-1,3-oxazole-4-carboxamide
1-methyl-1-[1-(4-methylpyridin-2-yl)propan-2-yl]-3-[2-(piperidin-1-ylmethyl)phenyl]urea
methyl 3-butanoyl-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[(1S)-1-(4-chlorophenyl)ethyl]-3-(1,5-dimethyl-1H-pyrazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
7-(cyclopropylmethyl)-N-[(2S)-2-hydroxypropyl]-8-oxo-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrrolidine-1-carboxamide
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzenesulfonamide
N-[3-(1H-indol-2-yl)phenyl]-1-(3-methylthiophene-2-carbonyl)piperidine-3-carboxamide
N-cyclopropyl-3-[1-(prop-2-ene-1-sulfonyl)piperidin-4-yl]propanamide
8-[(2,5-difluorophenyl)methyl]-3-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 2-[N-methyl-3-(2-methylphenyl)-3-phenylpropanamido]acetate
N-[2-(ethanesulfonyl)ethyl]-5-ethylpyrazolo[1,5-a]pyrimidin-7-amine
1-[1-benzyl-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-(thiophen-2-yl)butan-1-one
1-methyl-1-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-(1-methyl-1H-1,2,4-triazol-3-yl)urea
1-methyl-3-phenyl-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}-1H-pyrazole
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-(2H-1,3-benzodioxol-5-yl)-3-methyl-1-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(2-methoxyacetyl)-N-[3-(2-methylphenyl)phenyl]-1,4-diazepane-1-carboxamide
N-{3-[4-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-3-oxopropyl}methanesulfonamide
N-{3-[3-(4-fluorophenoxymethyl)piperidin-1-yl]-3-oxopropyl}-N-methylmethanesulfonamide
4-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-4-oxo-N-phenylbutanamide
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-1-(piperidin-1-yl)cyclohexane-1-carboxamide
N-(2-hydroxybutyl)-4-[(2-methoxyethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-5-hydroxypyrazine-2-carboxamide
6-{[2-methyl-2-(pyrrolidin-1-yl)propyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
1-(4-methanesulfonylphenyl)-5-methyl-1H-pyrazole-3-carboxylic acid
9-(3-amino-3-phenylpropanoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(3,5-dimethoxyphenyl)-2-{methyl[1-(pyrimidin-4-yl)ethyl]amino}acetamide