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6-[2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]pyridine-3-carboxamide
4-methyl-2-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
1-(2-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}phenyl)ethan-1-one
2-ethoxy-6-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
5-{3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}pyrazin-2-ol
ethyl 1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[({[1-(morpholin-4-yl)cyclohexyl]methyl}amino)methyl]-1H-pyrazole-4-carboxylate
N-(3-hydroxy-2,2-dimethylpropyl)-2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]acetamide
1-{3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}-2-(dimethyl-1,2-oxazol-4-yl)ethan-1-one
N-[(7-{[4-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]oxolane-3-carboxamide
6-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[(5-methylthiophen-2-yl)methyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
3-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-N,N-dimethyl-1H-1,2,4-triazol-5-amine
N-{3-[4-({2-[2-(trifluoromethyl)phenyl]ethyl}amino)piperidin-1-yl]phenyl}pyridine-4-carboxamide
2-[3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)propanamido]-2-methylpropanamide
N-({7-[3-(2-fluorophenyl)benzoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)propane-1-sulfonamide
(2R,3R)-3-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-{[5-(4-fluorophenyl)furan-2-yl]methyl}-2-(oxolan-3-yl)-1H-imidazole
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
methyl (2S)-2-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}formamido)-3-phenylpropanoate
2-(2H-1,3-benzodioxol-5-yl)-1-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
3-{1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(3-methoxyphenyl)-3-{1-[(5-methyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}propanamide
3-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}-N-(1,2,3-thiadiazol-5-yl)benzamide
1-(dimethylamino)-2-[4-(naphthalen-1-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-2-ol
N-(propan-2-yl)-2-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidin-4-amine
3-(4-phenoxybenzoyl)-1-(1,3-thiazole-4-carbonyl)piperidine
methyl 3-(5-ethyl-1,2-oxazole-3-carbonyl)-9-[2-(2-fluorophenyl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{2-[3-methyl-1-(naphthalen-1-yl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
3-acetyl-N-{3-[methyl(phenyl)amino]propyl}-1H-pyrazole-5-carboxamide
(2S)-2-amino-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-(1H-imidazol-4-yl)propanamide
N-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-N-[(1-methyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
3-methoxy-5-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
6-(2,5-dimethylfuran-3-yl)-N-(2-methoxybutyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-cyclooctyl-2-[(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)amino]acetamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[(2-ethoxy-2-oxoethyl)carbamoyl]piperidine-3-carboxylate
1-methyl-4-{1-[(4-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}piperazine
[(6-ethoxypyridin-3-yl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
1-[4-(pyrimidin-2-yl)piperazin-1-yl]-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
8-(3,4-dimethoxybenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-6-methylpyridine
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-1-(propan-2-yl)piperidine-3-carboxamide
(3R,4R)-1-(2,4-difluorobenzoyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-[(2-fluorophenyl)methyl]-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1H-1,2,3-triazole-4-carboxamide
6,7-dimethoxy-2-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1,2,3,4-tetrahydroisoquinoline
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-2-(2,3-dihydro-1H-indol-1-yl)ethan-1-one
N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(3-{pyrazolo[1,5-a]pyridin-7-yl}phenyl)methyl]propanamide
N-[(2R,3R)-1'-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
1-tert-butyl-5-(4-chloro-1-methyl-1H-pyrrol-2-yl)-3-methyl-1H-1,2,4-triazole
1-{[1-(2,3,5,6-tetramethylbenzoyl)pyrrolidin-2-yl]methyl}-1H-pyrazole