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N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]cyclohex-3-ene-1-carboxamide
1-[4-({[(3-chlorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(diethylamino)propan-2-ol
1-[(2,6-difluorophenyl)methyl]-4-ethyl-1,4-diazepan-5-one
2-[(1S,5R)-6-benzyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-cyclopropylpyridine-4-carboxamide
4-[4-(2-methoxyphenoxy)piperidin-1-yl]pyridine
2-{[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-4-methyl-1H-imidazole
2-{5-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
7-methyl-2-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
1-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
3-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-N,N-dimethylpyrazin-2-amine
1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-(pyridin-3-yl)piperidin-4-ol
N-(2-chloro-6-methylphenyl)-2-methyl-4-(2-methylpropyl)-3-oxopiperazine-1-carboxamide
(1S,4S)-2-{3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-2-azabicyclo[2.2.1]heptane
N-ethyl-3-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-4-{imidazo[1,2-b]pyridazin-6-yl}piperazine
1-cyclohexyl-N-[1-(naphthalen-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[2-(3,3-diphenylpiperidin-1-yl)-2-oxoethyl]pyrrolidin-2-one
N-({7-[2-(4-methoxyphenyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
1-[6-hydroxy-4-(4-methylpyrimidine-5-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
2-[4-(5-methyl-1H-indazole-3-carbonyl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
3,4-dimethoxy-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
3-{2-[cyclohexyl(methyl)amino]ethyl}-8-[(2R)-2-hydroxypropanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(furan-2-yl)-2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethane-1,2-dione
6-(cyclopropylmethoxy)-4-(dimethyl-1,3-thiazole-5-carbonyl)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
6-(2,6-dimethylpyrimidine-4-carbonyl)-3-(3-fluorophenyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
methyl (2S)-2-{[7-(2-methoxyacetamido)-1-methyl-2-phenyl-1H-1,3-benzodiazol-5-yl]formamido}-2-phenylacetate
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amine
1-[2-(4-chloro-2-methylphenoxy)ethyl]-4-(pyrrolidine-3-carbonyl)piperazine
1-{1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
4-(3-acetyl-1H-pyrazole-5-carbonyl)-6-(benzyloxy)-1-cyclohexyl-1,4-diazepan-2-one
3-(1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
N-[(2R,3R)-1'-[(5-chloro-2-hydroxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
1-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-3-(thiophen-2-yl)propan-1-one
N-methyl-N-(1,2-oxazol-5-ylmethyl)-4-oxo-3,4-dihydroquinazoline-2-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
2-(2-methoxyethoxy)-1-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
5-(3-fluorophenyl)-4-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-2-(trifluoromethyl)pyrimidine
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
1-[3-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)piperidin-1-yl]ethan-1-one
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-5-ethyl-1,3-oxazole-4-carboxamide
N-butyl-1-cyclopropyl-N-methyl-6-oxopiperidine-3-carboxamide
2-(furan-3-yl)-2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}acetic acid
(2E)-N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-3-(4-chlorophenyl)prop-2-enamide
N-cyclohexyl-4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
[(3R,5R)-5-[(dimethylamino)methyl]-1-(4-ethyl-5-methylthiophene-3-carbonyl)piperidin-3-yl]methanol
5-{[4-(azepane-1-carbonyl)-1,3-oxazol-2-yl]methoxy}-2-methyl-1,3-benzothiazole
(3S,7S,8aS)-7-{[(3-fluoro-4-methylphenyl)methyl]amino}-3-(1H-indol-3-ylmethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-[5-(4-cyclopentylpiperazin-1-yl)-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
2-benzyl-8-(morpholine-4-sulfonyl)-2,8-diazaspiro[4.5]decan-3-one
2-[(1H-indol-5-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid