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1-[4-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
4-(4-fluoro-2-methylphenoxy)-1-(2-methoxyacetyl)piperidine-4-carboxylic acid
N-(6-cyanopyridin-3-yl)-3-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}benzamide
(1S,3R)-3-amino-N-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}cyclopentane-1-carboxamide
1-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-2-(morpholin-3-yl)ethan-1-one
1-benzyl-4-[2-(methylsulfanyl)acetyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-{1-[(5-propylfuran-2-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
4-[(2-methyl-1,3-oxazol-4-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[(2-aminopyrimidin-5-yl)methyl]-4-(2-methylpropyl)-1,4-diazepan-6-ol
2,5-dimethyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)furan-3-carboxamide
6-methoxy-N-methyl-2-oxo-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-({8-[(2-methylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-4-(1H-pyrazol-1-yl)benzamide
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[3-(pyridin-3-yloxy)propyl]propanamide
N-{1-[1-(2,2-dimethylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
1-({4-methyl-5-[1-(piperidin-4-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
3-[2-(4-acetyl-1,4-diazepan-1-yl)-2-oxoethyl]-1-(cyclohexylmethyl)-3-phenylpyrrolidine-2,5-dione
[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl](methyl)[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amine
N-({8-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)benzamide
N-(1-methanesulfonylpiperidin-4-yl)-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
2-(4H-1,2,4-triazol-4-yl)-N-{[3-(trifluoromethoxy)phenyl]methyl}pyridine-4-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-4-[(pyridin-2-ylsulfanyl)methyl]benzamide
methyl 6-({[1-(4-methylpyridin-2-yl)propyl]carbamoyl}amino)-1,2,3,4-tetrahydroquinoline-1-carboxylate
1-methyl-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclohexane-1-carboxamide
(1R,5R)-N,N-dimethyl-6-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-(4-fluorophenyl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
benzyl 3-[1-(propan-2-yl)-1H-pyrazole-4-amido]pyrrolidine-1-carboxylate
dimethyl({[(1R,5S,6S)-3-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
4-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
(2S,4R)-4-[(4-fluorophenyl)sulfanyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-1-[(4-methylphenyl)methyl]pyrrolidine-2-carboxamide
N3-[(2,6-difluorophenyl)methyl]-N5-(2-methoxyethyl)-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-[(4-chlorophenyl)methyl]-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3-benzoxazole-5-carboxamide
(3R)-4-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]morpholine-3-carboxylic acid
methyl 4-(3-{[(4-fluorophenyl)formamido]methyl}piperidine-1-carbonyl)benzoate
2-methyl-N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
3-ethyl-1-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]piperazine
3-{imidazo[1,2-a]pyridine-2-carbonyl}-9-methoxy-N-methyl-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(3-chloro-4-fluorophenyl)-3-[1-(pyrimidin-2-ylmethyl)piperidin-4-yl]propanamide
(3R,4S)-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-4-phenylpyrrolidin-3-amine
5-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{[4-(1,3-benzothiazol-2-yl)-1,4-diazepan-1-yl]methyl}-3-hydroxy-1-methylpiperidin-2-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylbenzamide
2,4-dichloro-3-{[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidin-1-yl]methyl}phenol
2-[2-(1H-imidazol-4-yl)ethyl]-8-[2-(propan-2-ylsulfanyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]propan-1-one
N-[2-(2-fluorophenyl)-2-hydroxyethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
4-[2-(dimethylamino)acetamido]-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]benzamide
2-({[3-(difluoromethoxy)phenyl]methyl}amino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 3-cyclobutaneamido-1-[2-(pyridin-2-yl)ethyl]-5-[(thian-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N,2,3-trimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine