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N-cyclopropyl-1-{1-[(2,6-difluorophenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
6-(2-fluorophenyl)-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine
2-{[(3S,4S)-3-hydroxy-4-(morpholin-4-yl)pyrrolidin-1-yl]methyl}-5,8-dimethylquinolin-4-ol
N-(3-fluoro-2-methylphenyl)-2-(2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-4-(thiophen-2-yl)phenoxy)acetamide
5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1,2,3,4-tetrahydroisoquinoline
2-[5-(3-chloro-5-fluoro-4-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]acetamide
3-hydroxy-1-(3-phenylpropyl)-3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}piperidin-2-one
2-{[(1S,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}quinolin-4-ol
N-methyl-2-{4-[3-(1H-pyrazol-1-yl)phenyl]phenoxy}acetamide
N-[(3S,4R)-4-propyl-1-(5-propyl-1,2-oxazole-3-carbonyl)pyrrolidin-3-yl]methanesulfonamide
methyl 4-{[(2-{4-[(2-methylphenyl)carbamoyl]-1H-1,2,3-triazol-1-yl}ethyl)amino]methyl}benzoate
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-2-(5-methyl-1,2-oxazol-3-yl)piperidine
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[1-(pyridin-3-yl)propan-2-yl]amine
N-(2-hydroxyethyl)-N-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
4-methyl-2-phenyl-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazine
2-methyl-6-[1-(6-methylpyridazin-3-yl)piperidin-3-yl]pyrimidin-4-ol
2-[(3,4-dimethoxyphenyl)methyl]-6-(morpholine-4-carbonyl)-1,3-benzoxazole
1-methyl-N-(1-{7-[(2E)-2-methylbut-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)piperidine-4-carboxamide
3-methyl-1-propyl-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-4-carboxamide
N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
3-(2-methoxypyridin-3-yl)-5-methylpyridin-2-amine
2-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}benzoic acid
5-methyl-N-[(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-3-yl)methyl]-1,2-oxazole-3-carboxamide
methyl 6-(2-chlorobenzoyl)-2-(piperidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]morpholine-4-carboxamide
3-[(2-chlorophenyl)methyl]-9-methoxy-10-(thiomorpholine-4-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
3-(3-chlorophenoxymethyl)-5-(furan-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,4-dimethyl-2-oxopentanamide
3,5-dimethyl-N-[(3R)-pyrrolidin-3-yl]-1H-indole-2-carboxamide
1-{2-[1-cyclopentyl-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}-N,N-diethylpiperidine-4-carboxamide
N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-4-(1H-1,2,3,4-tetrazol-5-yloxy)aniline
3-[(2,4-dimethoxyphenyl)methyl]-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-(2-{[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amino}pyrimidin-4-yl)-2-ethoxybenzoic acid
2-[1-cyclopentyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-ethyl-N-(pyridin-4-ylmethyl)acetamide
5-chloro-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(pent-2-yn-1-yl)pyrrolidin-3-yl]pyridine-2-carboxamide
2-methoxy-N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)acetamide
3-[1-(4-chloro-2-methoxy-5-methylphenyl)-1H-imidazol-2-yl]pyridine
3-(1,4-diazepane-1-carbonyl)-N-[2-(pyridin-2-yl)ethyl]benzene-1-sulfonamide
2-(2H-1,3-benzodioxol-5-yl)-1-[7-(5-chloropyridin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
1-(oxolan-2-ylmethyl)-1-(pyridin-4-ylmethyl)-3-[4-(1H-1,2,4-triazol-1-yl)phenyl]urea
5-methyl-N-(morpholin-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
3-{[cyclopropyl(pyridin-3-ylmethyl)amino]methyl}-6,8-dimethyl-1,2-dihydroquinolin-2-one
1-{2-[3-(morpholin-4-yl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
2-[5-({[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]sulfanyl}methyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-1-yl]pyridine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3S)-3-(dimethylamino)azepan-1-yl]butan-1-one
N-{[8-(2,5-dimethoxybenzoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2-fluorobenzamide
1-(cyclopropanesulfonyl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid