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1-{4-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]phenyl}ethan-1-one
8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[4-(4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-2,5-dioxo-4-propylimidazolidin-4-yl}piperidine-1-carbonyl)phenyl]acetamide
1-(2,3-dimethylquinoxalin-6-yl)-3-[3-(2-ethyl-1H-imidazol-1-yl)propyl]urea
{1-[3-(1H-imidazol-2-yl)benzoyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)propanamide
N-[3-(1H-imidazol-5-yl)phenyl]-4-(oxolane-2-carbonyl)-1,4-diazepane-1-carboxamide
1-[4-(3-methylbutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-2-phenylethan-1-ol
1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-3-(3-fluoro-4-methoxybenzoyl)piperidine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]propanamide
2-(2-chlorophenoxy)-1-(7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
1-{[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidin-4-ol
4-{4-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}-2-methylbutan-2-ol
ethyl 4-(2-{4-[3-(2-methoxyphenyl)propanamido]-1H-pyrazol-1-yl}acetamido)piperidine-1-carboxylate
[(5-ethylpyridin-2-yl)methyl](methyl){[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2-(5-methyl-1H-pyrazol-1-yl)acetamide
2-({2-[(benzenesulfonyl)methyl]phenyl}methyl)-5-(dimethylamino)-2,3-dihydropyridazin-3-one
2-({1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidin-3-yl}formamido)-N-methylacetamide
ethyl 1-(5-methyl-1H-indazole-3-carbonyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
1-(adamantan-1-yl)-4-(1,3-thiazole-4-carbonyl)piperazine
2-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}benzoic acid
1-(2-chloro-4-fluoro-5-methylphenyl)-3-[(1-propyl-1H-imidazol-2-yl)methyl]urea
{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(thiophen-2-yl)ethyl]amine
N-(furan-2-ylmethyl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
N-(2,2-dimethyloxan-4-yl)-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[4-(trifluoromethyl)pyrimidin-2-yl]-decahydro-1,6-naphthyridin-2-one
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-[(2S)-oxolane-2-carbonyl]piperidine-4-carboxylic acid
1-{2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
1-(2-methoxyethyl)-8-[1-(methylsulfanyl)propan-2-yl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(2-methoxyacetyl)-N-[(3-phenoxyphenyl)methyl]piperidine-4-carboxamide
(1S,5R)-6-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
3-[5-(1H-imidazol-1-ylmethyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
1'-[5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carbonyl]spiro[indene-1,4'-piperidine]
[(2,5-dimethoxyphenyl)methyl]({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amine
14-(3,4-dimethylphenyl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2,5-dichloro-N-(2-oxo-2-{3-oxo-2,8-diazaspiro[4.5]decan-8-yl}ethyl)benzamide
N-{3-[methyl(phenyl)amino]propyl}-2-(morpholine-4-carbonyl)pyridin-4-amine
1,3-dimethyl-2,6-dioxo-N-{2-[(pyridin-3-yl)amino]ethyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(3aS,6aR)-5-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
7-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
(4aS,8aR)-1-(pyridin-3-ylmethyl)-6-(pyrimidin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
3-[2-(dimethylamino)ethyl]-5-{1-[2-(2-fluorophenyl)acetyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-2-methyl-4-(4-methylphenyl)piperazine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(4-fluorophenyl)methyl]piperidine-3,5-dicarboxamide
(3R,4S)-4-cyclopropyl-1-[4-(1H-pyrazol-3-yl)benzoyl]pyrrolidin-3-amine
1-[7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-(dimethylamino)ethan-1-one
5-ethyl-N-({3-methyl-7-[(2E)-4-methylpent-2-enoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,2-oxazole-3-carboxamide
1-(oxolan-2-ylmethyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
N-[(3S,4R)-4-(propan-2-yl)-1-(3,4,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-3-yl]acetamide