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N-(8-methylquinolin-5-yl)-4-(1H-pyrazol-3-yl)piperidine-1-carboxamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)acetamide
8-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2-[2-(dimethylamino)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
6-(2,5-dimethylphenyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
ethyl 4-{[(1R,2S)-2-(dimethyl-1,3-oxazole-4-amido)cyclobutyl]amino}piperidine-1-carboxylate
4-(1-methyl-1H-pyrazol-4-yl)-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrimidin-2-amine
1-(3-{[3-(dimethylamino)propyl](methyl)amino}piperidin-1-yl)-3-(2-methoxyphenyl)propan-1-one
3-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(2-ethylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[(2-methylprop-2-en-1-yl)amino]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]propanamide
(4aR,7aS)-1-[2-(4-ethoxypiperidin-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(2-ethoxyphenyl)methyl]-3-{2-[4-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
ethyl 1-(4-acetylbenzoyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
methyl 3-{[2-(2-methoxy-2-oxoethyl)-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl]methyl}benzoate
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-[3-(propan-2-yloxy)propyl]-1,3-oxazole-4-carboxamide
2-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-4H-chromen-4-one
3-[4-(2-ethoxyethyl)piperazine-1-carbonyl]-4,5,6-trimethyl-1,2-dihydropyridin-2-one
4-(4-methoxyphenoxy)-1-(2-methyloxane-2-carbonyl)piperidine
1-(furan-2-ylmethyl)-5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
9-(2,3-difluorobenzoyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(2S,3R)-2-amino-3-hydroxybutanoyl]-N-(2-methoxyethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
methyl 4-methoxy-3-{[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]amino}benzoate
3-[(benzylsulfamoyl)amino]-N-(pyridin-3-yl)benzamide
1-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-3-ol
(3S,4R)-3-(dimethylamino)-N-(furan-2-ylmethyl)-4-(4-methoxyphenyl)pyrrolidine-1-carboxamide
5-methoxy-2-[2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-1H-indole
N-(4-butanamido-3-methoxyphenyl)-1-(2-methylpropyl)-5-oxopyrrolidine-3-carboxamide
ethyl 4-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine-1-carboxylate
1-{3,9-diazaspiro[5.5]undecan-3-yl}-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
3-[ethyl({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)amino]-2,2-dimethylpropan-1-ol
1-(cyclohexylmethyl)-3-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-3-phenylpyrrolidine-2,5-dione
2-[2-({2-methyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)phenoxy]acetic acid
7-(cyclopropylmethyl)-6-(2-fluoro-4-methoxyphenyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(isoquinolin-5-ylmethyl)-N-methylacetamide
5-[(4-fluoro-3-methoxyphenyl)methyl]-5-{3-[4-(3-fluorophenoxy)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]acetamide
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
N'-[(3-methylphenyl)methyl]-N'-(propan-2-yl)pentanediamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-phenyl-1,2-oxazole-3-carboxamide
(3R,5S)-N-[3-(dimethylamino)propyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}piperidine-3-carboxamide
1-cyclohexyl-4-[3-(1-phenylethyl)-1,2-oxazole-5-carbonyl]piperazine
3-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1,2,5,6,7,8-hexahydroquinolin-2-one
4-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-6-methyl-1-[2-(methylsulfanyl)phenyl]piperazin-2-one
3-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chlorophenyl)urea
1-ethyl-3-(thiomorpholine-4-carbonyl)-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-({[(1-acetylpiperidin-4-yl)methyl]amino}methyl)-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
7-(cyclobutylmethyl)-2-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-2,7-diazaspiro[4.5]decan-6-one
6-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
3-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-3,9-diazaspiro[5.6]dodecan-10-one