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1-[4-(hydroxydiphenylmethyl)piperidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
3-{2-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}-1,3-thiazolidine-2,4-dione
1-{4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzoyl}piperidine
1-(2-cyclohexylethyl)-3-hydroxy-3-[({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amino)methyl]piperidin-2-one
1-(3-{[(adamantan-1-yl)amino]methyl}-7-methylquinolin-2-yl)piperidin-4-ol
(3S,4S)-1-[(3-methylthiophen-2-yl)methyl]-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}pyrrolidin-3-ol
2-[4-(4-phenylbenzenesulfonyl)morpholin-3-yl]acetic acid
2-[3-(3-methylpyrazin-2-yl)-1H-pyrazol-1-yl]-N-(1-propyl-1H-pyrazol-5-yl)acetamide
N-ethyl-N-[2-(4-methoxyphenoxy)ethyl]-4-(1H-1,2,4-triazol-5-yl)benzamide
N-cyclopropyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]imidazo[1,2-a]pyrimidine-2-carboxamide
3-[2-(dimethylamino)ethyl]-8-(2-fluoro-4-methylbenzoyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-benzyl-3-ethyl-1-(5-propylpyrimidin-4-yl)-1,4-diazepan-5-one
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-[3-(pyridin-4-yl)propyl]-5-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}[(1-ethyl-1H-pyrazol-4-yl)methyl]amine
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
4-(dimethoxy-1,3,5-triazin-2-yl)benzamide
2-(2,5-dimethoxyphenyl)-N-[1-(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)-2-phenylethyl]acetamide
8-cycloheptyl-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aR,6aS)-5-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-(4-chlorophenyl)-N-methyl-N-(oxolan-3-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{2-methyl-3-[(1,3-thiazol-2-yl)carbamoyl]phenyl}-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N-(3-{[(2,2-dimethylpropyl)amino]methyl}-5-(4-methylpiperazine-1-carbonyl)phenyl)acetamide
3-{2-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-3-(3-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-4-methyl-1,2,5-oxadiazole-3-carboxamide
4-ethyl-1-(3-phenylpropyl)-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S)-1-{3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanoyl}pyrrolidine-2-carboxamide
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]acetamide
1-{3-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-oxopropyl}piperidin-2-one
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(5-ethylfuran-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cyclopropyl-3-{1-[2-(4-methoxyphenoxy)acetyl]piperidin-3-yl}propanamide
N-[3-(methylsulfanyl)propyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
2-[2-oxo-4-(1-phenylcyclopentanecarbonyl)piperazin-1-yl]benzonitrile
1-(4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-diazepan-1-yl)-2-methoxyethan-1-one
5-cyclopropanecarbonyl-1'-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
15-methyl-12-(2-methylpiperidine-1-carbonyl)-9-(pyridin-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
methyl[(pentafluorophenyl)methyl](quinolin-6-ylmethyl)amine
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-[1-(quinoline-6-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
6-[4-methyl-3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]-2,3-dihydropyridazin-3-one
[4-(2-phenylethyl)-1-(quinolin-2-yl)piperidin-4-yl]methanol
{[2-(azocan-1-yl)pyridin-3-yl]methyl}(2,1,3-benzoxadiazol-5-ylmethyl)amine
1-(3-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}piperidin-1-yl)propan-1-one
(5S,9aS,9bS)-2-[(5-methylfuran-2-yl)methyl]-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]propanamide
(1S,5R)-6-(3-phenyl-1H-pyrazole-4-carbonyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
4-(4-methylbenzenesulfonyl)-7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-(dimethyl-1,2-oxazol-4-yl)acetamide
ethyl 4-{6-[(2,3-difluorophenyl)methyl]-6-azaspiro[2.5]octane-1-carbonyl}piperazine-1-carboxylate
1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
1-[4-(4-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)phenyl]ethan-1-one