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(2R,3S,6R)-3-phenyl-5-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
2-phenyl-1-[4-(1H-pyrazol-3-yl)phenyl]ethan-1-one
N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-4-(trifluoromethyl)pyrimidin-2-amine
N3-[(4-fluorophenyl)methyl]-1-(2-methoxyethyl)-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-cyclopropyl-1-(2,5-dichlorophenyl)-5-[2-(2-methyl-1H-imidazol-1-yl)propyl]-1H-1,2,4-triazole
2-methyl-N-(2-methylpropyl)-4-phenyl-N-(pyridin-2-ylmethyl)pyridine-3-carboxamide
(4aS,7aR)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(1-phenylethyl)-1,2-oxazole-5-carbonyl]piperidine
(1-{[methyl(quinolin-2-ylmethyl)amino]methyl}cyclopropyl)methanol
1-(4-{3-[(3-fluorophenyl)amino]piperidine-1-carbonyl}phenyl)ethan-1-one
N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
4-(2-methyl-1H-imidazol-1-yl)-1-{thieno[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
7-(2-methoxyacetamido)-N,1-dimethyl-N-[2-methyl-3-(pyrrolidin-1-yl)propyl]-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
1-methanesulfonyl-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazine
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-[(2R,3R)-1'-[(6-chloro-2H-chromen-3-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
9-(2-hydroxyacetyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
4-(2-methylpropanoyl)-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
3-[(1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}piperidin-4-yl)methyl]benzoic acid
(2S)-1-[2-(2,4-difluorophenoxy)acetyl]pyrrolidine-2-carboxamide
N-methyl-3-(1-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperidin-3-yl)-N-(1-methylpiperidin-4-yl)propanamide
1-[4-(2-ethoxyphenyl)piperazin-1-yl]-3-(oxolan-2-yl)propan-1-one
9-(4-fluoro-2-methylbenzoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(3,4,5-trimethoxyphenyl)benzonitrile
8-(2-fluoro-5-methylbenzenesulfonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-[2-(1H-pyrazol-4-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 4-(6-methyl-3-{[(2-methylpropyl)amino]methyl}quinolin-2-yl)piperazine-1-carboxylate
1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]piperidine-3-carboxamide
1-(2-methyl-1,3-thiazole-4-carbonyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-cyclopentyl-4-hydroxy-2-(pyridin-2-yl)-N-(thiophen-3-ylmethyl)pyrimidine-5-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,4,6-trimethylquinolin-2-amine
4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-N-(1-methylpiperidin-3-yl)pyrimidin-2-amine
3-(furan-2-ylmethyl)-1-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)urea
5-(4-chlorobenzoyl)-N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4,6-dimethyl-1-(2-{4-[2-(3-methylphenyl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}ethyl)-1,2-dihydropyrimidin-2-one
N2-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-N4-methylpyrimidine-2,4-diamine
2-cyclopropyl-8-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(oxolan-3-yl)-1,2-oxazole-3-carboxamide
2-(dimethylamino)-N-[5-({[3-(4-hydroxyphenyl)propyl]carbamoyl}amino)-2-methylphenyl]acetamide
1-ethyl-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-(piperidin-3-ylmethyl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}-1H-1,2,3-triazole-4-carboxamide
7-methyl-3-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzothiazole
5-{2-oxo-2-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-N,N-dimethylpiperidine-1-carboxamide
2-(5,5-dimethyl-2,4-dioxoimidazolidin-1-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
5-[2-(morpholin-3-yl)acetamido]pyridine-3-carboxylic acid
1-acetyl-N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}piperidine-4-carboxamide