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4-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-methyl-6-propylpyrimidine
1-(1-oxo-1,3-dihydro-2-benzofuran-5-yl)-3-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}urea
1-ethyl-N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)piperidine-2-carboxamide
(2E)-N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-3-(thiophen-2-yl)prop-2-enamide
5-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-yl](thiophen-2-yl)methanol
[1-(6-ethyl-2-methylquinoline-4-carbonyl)-3-[(4-fluorophenyl)methyl]piperidin-3-yl]methanol
4-(3-hydroxy-3-methylbutyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
5-ethyl-2-methyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}pyrimidin-4-amine
3-[4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]-1-methylpiperidine
methyl 3-[(3S,4R)-4-(dimethylamino)-1-[(4-ethoxyphenyl)methyl]piperidin-3-yl]propanoate
N-cyclopropyl-5-(dimethyl-1,3-thiazole-5-carbonyl)-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3R,4S)-4-propyl-1-(5-propyl-1,2-oxazole-3-carbonyl)pyrrolidin-3-amine
3-methoxy-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propan-1-one
7-(6,7-dimethoxy-4-methylquinolin-2-yl)-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 5-methyl-4-{1-oxa-8-azaspiro[4.5]decan-8-yl}thieno[2,3-d]pyrimidine-6-carboxylate
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
2-[2-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl]pyridine
3-{2-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}phenol
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
(4aR,7aS)-1-methyl-4-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-benzyl-N-(6-methoxypyridin-3-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-(1H-pyrazol-1-yl)benzamide
6-fluoro-4-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,2-dihydroquinolin-2-one
N4-[(1-methyl-1H-pyrazol-4-yl)methyl]-7-(oxolan-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
2-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-fluoropyridine
4-{1H-imidazo[4,5-b]pyridin-2-yl}-3-(3-methoxyphenyl)-1-phenyl-1H-pyrazole
1-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
N,2-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}furan-3-carboxamide
1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-{[7-(2,3-dimethyl-1H-indole-7-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-sulfonamide
ethyl 1-[1-(4-cyclopentaneamidophenyl)piperidin-4-yl]piperidine-3-carboxylate
1-[(2S,4R)-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]-1-[(2-fluorophenyl)methyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
4-[2-(4-fluorophenyl)piperidine-1-carbonyl]morpholine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[3-(1,2-oxazinan-2-yl)propanoyl]piperazin-2-one
{[5-(4-chlorophenyl)furan-2-yl]methyl}(methyl)({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
(3R,4R)-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-(hydroxymethyl)piperidin-3-ol
methyl 5-{[(4-methoxy-3-methylphenyl)methyl]amino}-3-(2-methoxyacetamido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-5-methylpiperidin-2-one
3-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-ol
2-[(2-{[3-(2,4-dimethylphenoxy)-2-hydroxypropyl]carbamoyl}phenyl)amino]acetic acid
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylimidazo[1,2-a]pyridine-6-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(isoquinolin-1-yl)-2,8-diazaspiro[4.5]decan-3-one
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(quinolin-6-ylmethyl)propanamide
2-butyl-5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-1,3-benzoxazole
(4aS,7aR)-4-ethyl-6,6-dioxo-N-[2-(thiophen-2-yl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(3S,9aR)-8-(3-methylbenzoyl)-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-(furan-3-ylmethyl)-1,4-diazepan-6-ol